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1'-(1,3-benzothiazole-6-carbonyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
1-ethyl-3-(propan-2-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
4-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]-1λ6-thiane-1,1-dione
3-[(2R,3R,6R)-5-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(1S,2S)-2-{4-[(2-methylquinolin-4-yl)methyl]piperazin-1-yl}cyclohexan-1-ol
4-cyclopentyl-3-{2-oxo-2-[4-(thiophen-2-ylmethyl)piperazin-1-yl]ethyl}piperazin-2-one
3-(4-{[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}-N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)benzamide
1-[2-({1,9-dioxaspiro[5.5]undecan-4-yl}amino)ethyl]-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-[(3-chlorophenyl)methyl]-4-(3-ethyl-1H-pyrazole-4-carbonyl)piperazine
3-[4-(thian-4-yl)piperazine-1-carbonyl]-1,2,3,4-tetrahydroisoquinolin-1-one
(4aS,7aR)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S)-1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-3-hydroxy-2-(methylamino)propan-1-one
3-(1-{[1-(9H-purin-6-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-1-ol
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-1-(diphenylmethyl)-N-methyl-1H-1,2,3-triazole-4-carboxamide
2-{2-[2-(dimethylamino)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}-N-methylpentanamide
1-[2-(4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1H-1,2,3-triazol-1-yl)ethyl]piperazine
5-acetyl-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)thiophene-2-carboxamide
4-(4-acetylpiperazin-1-yl)-2-[2-(3-methoxyphenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
1-{6-[4-(hydroxymethyl)-4-(2-phenoxyethyl)piperidin-1-yl]pyridin-3-yl}ethan-1-one
1-[(4-methoxyphenyl)methyl]-1-methyl-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
(3S,4S)-4-cyclopropyl-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}pyrrolidine-3-carboxylic acid
2,3,5-trimethyl-N-(2,2,2-trifluoroethyl)pyrazolo[1,5-a]pyrimidin-7-amine
2-(2-methylpropyl)-8-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,8-diazaspiro[4.5]decan-3-one
2-chloro-9-methyl-3-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)-4H-pyrido[1,2-a]pyrimidin-4-one
N-[(3S,4R)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]amine
1-[(4-fluorophenyl)methyl]-4-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1,4-diazepane
2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-(oxolan-2-ylmethyl)acetamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(2-methylpropanoyl)piperidine-3-carboxylate
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
2-(4-cyclohexylpiperazin-1-yl)-2-(4-hydroxyphenyl)acetic acid
(3R,5S)-5-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidin-3-ol
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]benzonitrile
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-(cyclohex-3-en-1-ylmethyl)piperidine-4-carboxamide
3-[5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-5-[2-(piperidin-2-yl)ethyl]phenol
5-ethyl-2-[1-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1H-imidazol-2-yl]pyridine
5-(1-{[4-(3-hydroxy-3-methylbut-1-yn-1-yl)phenyl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
ethyl 4-[2-(1H-pyrazol-4-yl)quinoline-4-carbonyl]piperazine-1-carboxylate
N-{2-[3-(ethylsulfanyl)-5-oxo-4,5-dihydro-1,2,4-triazin-6-yl]phenyl}-2,3-dihydro-1-benzofuran-7-carboxamide
5-{2-[5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-3-(propan-2-yl)-1,2,4-oxadiazole
[1-(2-methoxyphenyl)ethyl](methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
(3aS,6aS)-2-(2-hydroxyethyl)-5-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3R,4S)-1-[2-methyl-2-(morpholin-4-yl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
4-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-1-benzyl-4-phenylpiperidine
1-(2-methoxyphenyl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)-1H-pyrazole-4-carboxamide