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(1s,4s)-4-({ethyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)cyclohexan-1-amine
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1,4-diazepan-6-ol
1-{2-[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)amino]-4-methylpyrimidin-5-yl}ethan-1-one
1-methyl-N-[1-(morpholin-4-ylmethyl)cyclopentyl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-(3-fluorophenyl)-3-{[methyl(prop-2-en-1-yl)amino]methyl}benzamide
3-{[3-ethyl-1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
4-chloro-N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}benzamide
methyl 3-(cyclobutylmethoxy)-5-[(3R)-3-methylpiperazine-1-carbonyl]benzoate
2-(4-ethyl-2-methyl-1,3-thiazol-5-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[2-(4-fluorophenyl)-2-hydroxyethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
[(4aS,8aR)-6-(3-phenylpropyl)-decahydro-1,6-naphthyridin-4a-yl]methanol
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}-5-[(propan-2-yl)sulfamoyl]benzamide
1-[3-(2-methylphenoxy)azetidin-1-yl]-2-(morpholin-3-yl)ethan-1-one
(3S,4S)-1-{[4-(2-fluorophenyl)phenyl]methyl}-4-(morpholin-4-yl)pyrrolidin-3-ol
N-methyl-2-[(2-methylprop-2-en-1-yl)oxy]-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}benzamide
1-[(3-chlorophenyl)methyl]-5-[1-(1H-imidazol-1-ylmethyl)cyclopropyl]-3-(2-methoxyethyl)-1H-1,2,4-triazole
N-(4-{1-[(1-hydroxycyclohexyl)methyl]-1H-imidazol-2-yl}phenyl)acetamide
3-[(3-fluorophenyl)methyl]-5-{[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,2,4-oxadiazole
N-ethyl-N-(oxan-4-ylmethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
4-ethyl-1-methyl-3-{1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({[(cyclooctylcarbamoyl)methyl]amino}methyl)-N-methylbenzamide
1-[(3R,4S)-3-(dimethylamino)-4-propylpyrrolidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
2-methyl-1-(pyrimidin-2-ylmethyl)-1,4-dihydroquinolin-4-one
ethyl 4-({[(1-cyclopentylpiperidin-4-yl)methyl](oxolan-2-ylmethyl)amino}methyl)-1H-pyrazole-3-carboxylate
2-(2-{[(3S)-3-(dimethylamino)azepan-1-yl]methyl}phenoxy)-1-(piperidin-1-yl)ethan-1-one
propan-2-yl 2-chloro-5-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}carbamoyl)amino]benzoate
4-(1-ethyl-1H-imidazol-2-yl)-1-[2-(4-fluorophenyl)benzoyl]piperidine
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-5-(2,4-dimethoxyphenyl)-1,2,4-triazin-3-amine
5-cyclohexaneamido-N-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carboxamide
2-{[(3-methylthiophen-2-yl)methyl]amino}-N-[2-(pyridin-3-ylformamido)ethyl]benzamide
N-{[5-(3-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
N3-{[3-(difluoromethoxy)phenyl]methyl}-N1,N1-dimethylpiperidine-1,3-dicarboxamide
2-(dimethylamino)-1-{5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethan-1-one
2-(2,6-dimethoxypyridin-3-yl)-2-[4-(furan-2-carbonyl)piperazin-1-yl]acetic acid
2-{[(3-cyano-2-methoxypyridin-4-yl)amino]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-(2-chloro-6-fluorophenyl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-6-[4-(morpholin-4-yl)piperidine-1-carbonyl]thieno[2,3-d]pyrimidin-4-amine
1-(2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-cyclopentyl-1H-1,2,4-triazol-5-yl}ethyl)-1H-1,2,3,4-tetrazole
(2S,4R)-4-amino-N-ethyl-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]pyrrolidine-2-carboxamide
6-methyl-2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}pyridine-3-carbonitrile
N-[3-({[(3-phenoxyphenyl)methyl]amino}methyl)-5-(pyrrolidine-1-carbonyl)phenyl]acetamide
1-methyl-2-[1-(propane-2-sulfonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
4-(benzyloxy)-1-(1,2-oxazole-5-carbonyl)piperidine
1-cyclohexyl-4-{2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetyl}piperazin-2-one
methyl 9-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]-7-oxo-3-(3-phenylprop-2-ynoyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(3-fluorophenoxy)-1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]ethan-1-one
dimethyl(2-{2-[1-(naphthalene-1-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
1-(2-phenylethyl)-4-[(quinolin-8-ylmethyl)amino]pyrrolidin-2-one
1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-4-(1,3-thiazol-2-yl)piperazine
(2S,4S)-4-amino-N,N-diethyl-1-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]pyrrolidine-2-carboxamide