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5-(oxolan-2-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}thiophene-2-carboxamide
4-{[(1S,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-2,1,3-benzoxadiazole
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)oxane-4-carboxamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(4-methyl-1H-imidazole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-[2-(2-methylphenyl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
2-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1H-indole
2-fluoro-5-[2-(quinolin-4-yl)-1H-imidazol-1-yl]benzonitrile
N-cyclopentyl-N-{[4-methoxy-3-(propan-2-yloxy)phenyl]methyl}-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
2-{4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-N-(2-phenylethyl)piperidine-4-carboxamide
methyl 1-{2-hydroxy-3-[3-(piperidin-1-ylmethyl)phenoxy]propyl}piperidine-4-carboxylate
4-{2-azaspiro[4.4]nonane-2-carbonyl}-5,7-dimethyl-2-(1H-pyrazol-4-yl)quinoline
(1R,5R)-3-cyclobutanecarbonyl-6-[(2,4-difluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-{2-methylimidazo[1,2-a]pyridin-3-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
3-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-9-methyl-3,9-diazaspiro[5.6]dodecane
{[8-methyl-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}[(3,4,5-trimethoxyphenyl)methyl]amine
7-[(2-fluorophenyl)methyl]-2-(pyridine-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-methylbut-2-enamide
4-(1H-imidazol-1-yl)-1-(2-methyl-6-propylpyrimidin-4-yl)piperidine-4-carboxylic acid
2-[(3S,4R)-4-amino-1-(trimethylpyrimidin-4-yl)pyrrolidin-3-yl]ethan-1-ol
2-(1-cyclopentyl-4-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl)ethan-1-ol
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-ol
4-(6-aminopyrimidin-4-yl)-2,2-diphenylbutanenitrile
N3-[2-(3-fluorophenyl)ethyl]-4-oxo-1-(oxolan-2-ylmethyl)-N5-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
benzyl(methyl)({3-[4-(pyridin-2-yl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methyl)amine
N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-{5-[1-(furan-2-ylmethyl)piperidin-4-yl]-1,2,4-oxadiazol-3-yl}-6-methylpyridazine
3-chloro-6-[2-(morpholin-4-ylmethyl)phenyl]pyrazolo[1,5-a]pyrimidine-2-carboxylic acid
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}cyclopropanamine
3-methyl-4-({[1-(1-methyl-1H-pyrazol-5-yl)propyl]carbamoyl}amino)-N-propylbenzamide
2-{4-[2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carbonyl]piperazin-1-yl}ethan-1-ol
N-(3-cyanophenyl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-(azocan-1-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]propanamide
2-(pyrazin-2-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
(cyclobutylmethyl)({[5-methyl-2-(thiophen-3-yl)-1,3-oxazol-4-yl]methyl})(oxolan-2-ylmethyl)amine
5-[5-(2H-1,2,3-benzotriazol-2-ylmethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
2-{4-[(5-methylfuran-2-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-{1-[2-methoxy-2-(thiophen-2-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-1,3-thiazole
1-(2,2-dimethylpropyl)-3-hydroxy-3-{[(propan-2-yl)amino]methyl}piperidin-2-one
methyl (2R,4S)-4-hydroxy-1-(isoquinoline-5-carbonyl)piperidine-2-carboxylate
methyl 5-(cyclohexylamino)-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(1S,3R)-3-{1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}cyclohexan-1-amine
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2-(morpholin-4-yl)ethyl]-1H-pyrazole-4-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-(benzylamino)-1-[(4-chlorophenyl)methyl]pyrrolidine-2-carboxamide
3-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine-1-carbonyl}-2-(methylsulfanyl)pyridine
N-(2,3-dihydro-1H-inden-1-yl)-6-(morpholin-4-yl)pyrimidin-4-amine
1-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}piperidin-3-ol
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide