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4-{2-[(2-methylpyrimidin-4-yl)oxy]hex-5-en-1-yl}-1,4-oxazepane
(1S,2S)-N2-{1-[2-(dimethylamino)-6-methylpyrimidin-4-yl]piperidin-4-yl}-2,3-dihydro-1H-indene-1,2-diamine
2-butyl-8-(3-phenyl-1,2-oxazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
5-cyclopropanecarbonyl-1'-(2,5-dimethylfuran-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-chloro-1-methyl-3-{[2-(5-methyl-1,2-oxazol-3-yl)pyrrolidin-1-yl]methyl}-1H-indazole
5-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
(1S,5R)-3-[2-(1H-imidazol-1-yl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(ethoxymethyl)-N-[2-(4-methyl-1H-pyrazol-1-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{4-[7-(hydroxymethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]piperidin-1-yl}acetamide
2-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}ethan-1-one
3-[1-(2-aminopyridine-4-carbonyl)piperidin-3-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
6-amino-N-[(1-benzyl-1H-pyrazol-4-yl)methyl]pyridine-3-carboxamide
4-{[1-(1-acetylpiperidin-4-yl)piperidin-4-yl]oxy}-3-chloro-N-(2-methoxyethyl)benzamide
methyl 2-[3-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)-1H-indol-1-yl]acetate
1-({5-[(4-ethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
N-{[7-chloro-2-(2,5-dimethoxyphenyl)quinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]furan-3-carboxamide
3-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-1-propyl-1H-pyrazole-4-carboxamide
1'-[(1-ethyl-1H-pyrazol-4-yl)sulfonyl]-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-[2-(4-fluorophenyl)ethyl]-1-(1,3-thiazole-4-carbonyl)piperidine
4-{[2-(1-methanesulfonylpiperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
(1S,4S)-2-(3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzoyl)-2-azabicyclo[2.2.1]heptane
7-chloro-3,5-dimethyl-N-[2-(oxan-2-yl)ethyl]-1-benzofuran-2-carboxamide
6-methoxy-3-[1-phenyl-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,4-dihydroquinolin-4-one
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-(dimethylamino)-8-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-{1-[1-(4-methylphenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
4-[(4-methyl-1H-pyrazol-1-yl)methyl]-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
2-(1,3-benzothiazol-2-ylmethyl)-4-{4-[(2,6-difluorophenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
ethyl 4-{1-ethyl-2,4-dioxo-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decan-8-yl}piperidine-1-carboxylate
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(1-hydroxy-2-methylpropan-2-yl)amino]pyridine-3-carboxamide
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-3-(1-methylpiperidin-3-yl)propanamide
1-[(1-ethyl-1H-imidazol-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-3-(methoxymethyl)piperidine
2,5-dimethyl-3-(4-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}piperazin-1-yl)pyrazine
N-[3-(tert-butylcarbamoyl)-2-methylphenyl]-1H-1,2,4-triazole-5-carboxamide
1-(1H-imidazol-4-ylmethyl)-3-(4-phenyl-1H-pyrazol-5-yl)piperidine
2-[3-(4-hydroxyphenyl)benzoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-phenoxybutan-1-one
1-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1,2-dihydroquinolin-2-one
(3aS,6aS)-2-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(4-fluorophenyl)urea
1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
4-({3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}methyl)-2,1,3-benzoxadiazole
3,3-dimethyl-1-[7-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]butan-1-one
N-[(4-chlorophenyl)(pyridin-4-yl)methyl]-2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
methyl 3-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-oxo-9-[2-(thiophen-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1S,5R)-3-[(2,3-difluoro-6-methoxyphenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(2-ethoxy-5-{[2-(4-methyl-1,2,5-oxadiazol-3-yl)pyrrolidin-1-yl]methyl}phenyl)methyl acetate
1-(4-fluorophenyl)-4-(5-phenyl-1,2,4-oxadiazol-3-yl)-1,4-diazepane
5-methoxy-2-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-1,4-dihydropyridin-4-one