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N-{2-chloro-5-[(propan-2-yl)carbamoyl]phenyl}-3-(dimethylamino)pyrrolidine-1-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-5-[4-hydroxy-1-(2-methylbutyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
2-(4-{[methyl(1,3-thiazol-2-ylmethyl)amino]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
2-[(2-methoxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]acetic acid
5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]-2-(1H-pyrrol-2-yl)pyridine
1'-[1-(4-methylquinazolin-2-yl)piperidine-4-carbonyl]spiro[indene-1,4'-piperidine]
5-(2-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
2-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]pyridin-3-ol
2-cyclopropanecarbonyl-8-(morpholine-4-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
5-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-N-ethyl-4-methyl-1,3-thiazol-2-amine
2-[2-({methyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)phenyl]-6-propyl-3,4-dihydropyrimidin-4-one
N-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-N-[(4-ethoxyphenyl)methyl]cyclopropanamine
2-(4-chloro-2-methylphenoxy)-1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}ethan-1-one
N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[3-(trifluoromethyl)phenyl]acetamide
1-(2-phenylpyrrolidin-1-yl)-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
(4aS,8aR)-6-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
4-{[1-(carboxymethyl)cyclohexyl]amino}pyrimidine-5-carboxylic acid
3-{3-[3-(2-methyl-1,3-benzoxazol-5-yl)phenyl]-1H-pyrazol-1-yl}propan-1-ol
N-[(2-fluorophenyl)methyl]-3-(4-methylpiperazine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(2-aminoethyl)-3-{[1-(4-fluorophenyl)propyl]sulfamoyl}benzamide
N-cyclopentyl-1-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]furan-2-carboxamide
N-ethyl-5-(2-ethylpiperidine-1-carbonyl)-1-[(3-methoxyphenyl)methyl]-N-(2-methylprop-2-en-1-yl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1-(9H-purin-6-yl)-N-{[3-(pyrazin-2-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-4-amine
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
2-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-{[4-(3-fluorophenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-1H-pyrazole-3-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-N-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]pyrrolidine-1-carboxamide
2-(6-aminopyridin-3-yl)-2-{spiro[indene-1,4'-piperidine]-1'-yl}acetic acid
1,9-dimethyl-4-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
1-[1-(6-aminopyridine-3-carbonyl)piperidin-4-yl]-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
2-amino-4-[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]-7-methyl-5H,7H-furo[3,4-b]pyridine-3-carbonitrile
2-{5-[1-(oxolan-3-yl)-4-phenyl-1H-imidazol-5-yl]furan-2-yl}benzonitrile
methyl N-[4-(morpholin-4-yl)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]carbamate
2-(2-hydroxyethyl)-9-[4-(trifluoromethyl)pyrimidin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
dimethyl(3-{2-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1H-imidazol-1-yl}propyl)amine
2-methyl-5-[4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N-[3-(cyclohexylsulfanyl)propyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[(4-chlorophenyl)methyl]-N-(3-hydroxypropyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
6-({2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}carbonyl)-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1R,5S,6R)-3-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxylic acid
7-(6-phenylpyridine-2-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
2-(3-{[2-(dimethylamino)-4-methylpyrimidin-5-yl]formamido}propanamido)acetic acid
5-(2-fluorophenyl)-N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}({[4-(methylsulfanyl)phenyl]methyl})amine
1-{[2-(8-methoxyquinolin-2-yl)phenyl]methyl}piperidin-4-one
1-(furan-2-ylmethyl)-4-{[1,2,4]triazolo[4,3-a]pyridine-7-carbonyl}-1,4-diazepan-6-ol
8-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-1-oxa-8-azaspiro[4.6]undecane