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N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
2-[4-(pyridin-3-ylmethyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
dimethyl({5-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]thiophen-3-yl}methyl)amine
2-{4-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]morpholin-3-yl}-N-(3,5-dimethylphenyl)acetamide
2-methyl-1-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]-1,4-diazepan-5-one
(3S)-3-[(benzylsulfamoyl)amino]azepan-2-one
({5-[(4-chlorophenyl)sulfanyl]furan-2-yl}methyl)[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-1-azabicyclo[2.2.2]octan-3-amine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,3-oxazole-4-carboxamide
(2S)-1-[2-(1H-imidazol-2-yl)ethyl]-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
1-{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
(2S,4R)-4-amino-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-1-[3-(2-oxopyrrolidin-1-yl)phenyl]urea
ethyl 4-{4-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]benzoyl}piperazine-1-carboxylate
(2S,4S)-4-amino-1-{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}-N-ethylpyrrolidine-2-carboxamide
1-cyclopentyl-N3-[3-(dimethylamino)-2,2-dimethylpropyl]-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
8-[4-(4-fluorophenyl)-4-oxobutyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
3-[4-(2-phenylethyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
4-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-3-methyl-1-[(3-methylphenyl)methyl]piperazin-2-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-3-(1,2-oxazolidin-2-yl)-N-(pyridin-3-ylmethyl)propanamide
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-3-(5-methylfuran-2-yl)-1H-pyrazole-5-carboxamide
6-methoxy-3-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-1,2-dihydroquinolin-2-one
2-(6-methoxynaphthalen-2-yl)-4-(6-methoxypyrimidin-4-yl)morpholine
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-2-(oxan-4-yl)acetamide
N-{[3-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-sulfonamide
3-cyclopropyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1H-pyrazole-5-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-(3-methyl-3-phenylpiperidin-1-yl)ethan-1-one
(1S,4S)-2-(2-fluorophenyl)-5-[(5-methylfuran-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
(4aR,7aS)-N,N-dimethyl-4-[2-(methylamino)-1,3-thiazole-4-carbonyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-2-(1-propylpiperidin-4-yl)acetamide
(2,3-dihydro-1-benzofuran-5-ylmethyl)[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amine
{1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidin-4-yl}(thiophen-2-yl)methanol
2-{3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]piperidin-1-yl}acetamide
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-(5-propyl-1,2-oxazole-3-carbonyl)piperidine
3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]propanamide
4-methyl-5-(2-{4-phenyl-5-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H-imidazol-1-yl}ethyl)-1,3-thiazole
4-(pyridin-3-ylmethyl)-7-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[4-(3-methoxypyrrolidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
ethyl 1-(7-chloroquinolin-4-yl)-5-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
1-[2-methoxy-5-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
7-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-2-oxa-7-azaspiro[4.5]decane
5-chloro-N-[2-(2,4-dimethylphenoxy)ethyl]-N-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
4'-[(6-methylpyridin-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
{3-[(2-aminopyridin-3-yl)methyl]-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
N-cyclopropyl-1-{1-[(2,5-dimethylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
(1R,2S)-2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)cyclopentane-1-carboxamide
N-methyl-5-(propan-2-yl)-N-(quinoxalin-2-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine