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{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
N-ethyl-2-(4-fluorophenyl)-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-{1-[1-(2-fluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylthiophene-3-carboxamide
N-(heptan-4-yl)piperidin-4-amine
N-[(2-methylphenyl)methyl]-2-[2-(2-oxopyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
N-[(1S,2R)-2-aminocyclobutyl]-7-chloro-1-cyclopropyl-6-fluoro-4-oxo-1,4-dihydroquinoline-3-carboxamide
1-(5-ethyl-1,3,4-thiadiazol-2-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
8-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
5-{[(3R,4S)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-N,N-dimethylfuran-2-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-(pyridin-3-yl)propanamide
N-(1-{1-[(4-ethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-fluorobenzamide
2-(dimethylamino)-N,4-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrimidine-5-carboxamide
1-(1H-imidazol-2-ylmethyl)-3-(methanesulfonylmethyl)piperidine
1-tert-butyl-N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-ethyl-4-{5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1-methylpiperazin-2-one
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-5-methylpiperidin-2-one
4-{1-[(4-methoxyphenyl)methyl]-1H-1,2,4-triazol-5-yl}-1λ6-thiane-1,1-dione
1-[4-phenyl-1-(thiophene-3-sulfonyl)piperidin-4-yl]ethan-1-one
3-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]-N-(thiophen-2-ylmethyl)propanamide
[3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propyl]({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
N-[(3S,5S,9S)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]-4-ethylbenzamide
N-[(2-aminopyridin-3-yl)methyl]-2-methyl-6-(piperidin-4-yl)pyrimidin-4-amine
4-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-2-[1-(thiophen-2-yl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[2-(dimethylamino)ethyl]-5-(3-hydroxy-4-methylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(7-chloro-1-methyl-1H-indole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-(2-{3-[3-methyl-7-(pyrimidin-2-yl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]-1,2,4-oxadiazol-5-yl}ethyl)acetamide
N-({3-methyl-7-[4-(piperidin-1-yl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)thiophene-3-carboxamide
5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-{2-[4-(trifluoromethyl)phenyl]-1,3-thiazole-4-carbonyl}thiomorpholine
1-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
3-(carbamoylmethoxy)-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]benzamide
N-(1-{7-[(5-ethylfuran-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
N-(1-{1-[(2R)-2-amino-4-methylpentanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
2-[5-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
3-methyl-4-[1-(1-phenylethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1-(prop-2-en-1-yl)-1H-pyrazole
1-(2,6-difluorobenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
3-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-1H-indazole
ethyl 2-[(2-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenyl)amino]acetate
2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
2-(4-fluoro-2-methoxyphenyl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]acetic acid
N-({1-[(2-methylpyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)cyclopropanesulfonamide
5-(azocan-1-yl)-1-ethyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
(1-{[1-(8-methoxyquinolin-2-yl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methanol
7-(cyclobutylmethyl)-2-(5-methoxy-4-oxo-4H-pyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]-1-(1H-imidazol-2-ylmethyl)piperidine
5-(3-chlorophenoxymethyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]cyclopropanecarboxamide
N3-[(2-fluorophenyl)methyl]-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-[1-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-4-phenyl-1H-imidazol-5-yl]pyridine