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{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}({[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl})amine
7-cyclohexyl-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-{3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-7-yl}-2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]ethan-1-one
N-[2-(dimethylamino)ethyl]-3-[1-(pyridine-3-sulfonyl)piperidin-4-yl]propanamide
1-{1-[(1-ethyl-1H-indol-3-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
5-(1H-indazol-1-yl)-3-methylpyridin-2-amine
2-{[1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
2-amino-1-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]-2-methylpropan-1-one
2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-4-oxo-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
5-propyl-N-(pyridin-3-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-oxazole-3-carboxamide
2-[(5,6-dimethyl-1H-1,3-benzodiazol-1-yl)methyl]-6-(piperidin-3-yl)-3,4-dihydropyrimidin-4-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-methoxy-4-(prop-2-en-1-yl)piperidine
3-(4-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-3-yl}pyridin-2-yl)phenol
1-[2-(2-hydroxyethoxy)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(1-{1-[(2,4-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
3-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N-(thiophen-2-ylmethyl)propanamide
N-[2-(pyridin-2-ylsulfanyl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-(6-chloropyridin-3-yl)-3-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]urea
2-ethyl-6-methyl-4-oxo-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}-1-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3-carboxamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}[1-(pyridin-4-yl)propyl]amine
N-methyl-4-(4-methylphenyl)-5-(pyridin-4-yl)-N-(pyrimidin-4-ylmethyl)pyrimidin-2-amine
(2R,3R)-3-amino-1'-(quinoline-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
{3-[(2,4-difluorophenyl)methyl]-1-[4-(methylamino)pyrimidin-2-yl]piperidin-3-yl}methanol
methyl 2-(5-methyl-2-{[2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)benzoate
2-(3-methoxyphenoxy)-1-[3-(2-methoxyphenoxy)azetidin-1-yl]propan-1-one
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
N-methyl-3-(1H-pyrazol-1-yl)-N-(1H-pyrazol-5-ylmethyl)benzamide
2-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-(1-{4-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]phenyl}ethyl)morpholine
4-{4-[2-(4-chloro-2-methylphenoxy)acetyl]piperazin-1-yl}-2-[2-(4-fluorophenyl)ethyl]-2,3-dihydro-1H-isoindole-1,3-dione
4-{2-methyl-6-[1-(2-propoxyethyl)piperidin-4-yl]pyrimidin-4-yl}morpholine
8-[2-(trifluoromethyl)morpholine-4-carbonyl]-1,2,3,4-tetrahydroquinoline
N-methyl-4-(piperidin-3-yl)-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}benzamide
5-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-N-phenylpyrimidin-2-amine
4-({[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-1,3-thiazol-2-amine
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(morpholin-4-yl)propanamide
6-fluoro-2-oxo-N-(1,3-thiazol-2-ylmethyl)-1,2-dihydroquinoline-4-carboxamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-[4-(1H-1,2,4-triazol-1-yl)phenoxymethyl]-1,2-oxazole-3-carboxamide
1-(4-ethoxy-2-fluorophenyl)-3-(2-methoxyethyl)-3-[(5-methylthiophen-2-yl)methyl]urea
2-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]pyrazine
(2R,5R)-1-({5-cyclopentyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5-dimethyl-4-(prop-2-en-1-yl)piperazine
(3S,7S)-5-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[2-(oxan-2-yl)ethyl]pyridin-2-amine
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-(4-methyl-1,4-diazepan-1-yl)propan-1-one
[2-(3-fluorophenyl)ethyl][(8-methyl-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}quinolin-3-yl)methyl]amine
4-methyl-2-(propan-2-yl)-5-[3-(pyridin-4-yl)azetidine-1-carbonyl]pyrimidine
(3S,4S)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide