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1-[(2-phenyl-1H-imidazol-4-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
3-methyl-4-[3-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]oxolan-2-one
8-({3-[(dimethylamino)methyl]phenyl}methyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
1-[1-(2-cyclopentylacetyl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
6-ethyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2,3-dihydro-1H-inden-1-yl)-1-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]ethan-1-one
(3S,9aR)-8-(4-methoxybenzoyl)-3-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(2-{4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)azepan-2-one
N,N-dimethyl-2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
[(dimethyl-1,2-oxazol-4-yl)methyl][1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amine
1-[(4-ethylphenyl)methyl]-5-[(2-methyl-1H-imidazol-1-yl)methyl]-1H-1,2,4-triazole
N-[1-(hydroxymethyl)cycloheptyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-{3-methyl-4-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}acetamide
N-ethyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-2-methanesulfonylethan-1-one
3-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-methylpropanamide
6-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carbonyl)pyridin-2-amine
8-(4-aminopyrimidin-2-yl)-3-[3-(4-ethylpiperazin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidine-4-carbonyl)thiomorpholine
2-(2,3-dihydro-1H-inden-1-yl)-N-(1,1-dioxo-1λ6-thian-4-yl)-N-methylacetamide
methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl][3-(methylsulfanyl)butyl]amine
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
8-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
10-(3-hydroxypiperidine-1-carbonyl)-9-methoxy-3-[(5-methylthiophen-2-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
(1S,5R)-3-(1H-indol-5-ylmethyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(3-chlorophenyl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-{[benzyl(methyl)amino]methyl}-N-cyclobutyl-1,2-oxazole-3-carboxamide
ethyl 1-[1-(dimethylcarbamoyl)piperidine-4-carbonyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1-hydroxy-3-methylbutan-2-yl)-1,3-oxazole-4-carboxamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(pyridin-2-yl)propanamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
4-[(1-{2-[4-(hydroxymethyl)phenyl]acetyl}pyrrolidin-3-yl)methyl]benzoic acid
4-[(3R,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
N-[(2S,4R,6S)-2-(2,1,3-benzothiadiazol-4-yl)-6-benzyloxan-4-yl]acetamide
4-(2-{3-[2-(methylsulfanyl)ethyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl}propan-2-yl)morpholine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-(5-methyl-1-propyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-[2-(2,4-difluorophenyl)ethyl]-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
4-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]-2-(trifluoromethyl)morpholine
6-tert-butyl-N-{[(2R)-1-ethylpyrrolidin-2-yl]methyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2R,3S,6R)-3-(4-methylphenyl)-5-(4-methylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}-N-propylpyrimidin-2-amine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(methylamino)pyrimidine-5-carboxamide
6-amino-2-[2-({5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}amino)ethyl]pyrimidin-4-ol
N-[2-(3,4-dimethylphenoxy)ethyl]imidazo[1,2-a]pyrimidine-2-carboxamide
1-[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
1-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
N-[2-(methylsulfanyl)ethyl]-5-[1-(thiophen-3-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
4-{6-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}morpholine
2-[2-(pyridin-2-yl)piperidine-1-carbonyl]-4-(1H-1,2,3,4-tetrazol-1-yl)phenol