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2-({4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]piperidin-1-yl}methyl)pyridine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-6-methylpyridazin-3-amine
2-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
(3S,4S)-1-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-cyclopentyl-N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)acetamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-5-methyl-1-propyl-1H-pyrazole
4-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-methylthieno[3,2-d]pyrimidine
3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-propyl-1,2,4-oxadiazole
5-chloro-2-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}pyrimidine
4-(3-chloro-4-methoxyphenyl)-2-methyl-1H-imidazole
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-5-fluoro-4-methoxypyrimidine
N-{2-cyclobutyl-1-methyl-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-7-yl}oxolane-2-carboxamide
N-cycloheptyl-3-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]propanamide
3-{[1-(quinolin-2-ylmethyl)pyrrolidin-3-yl]methyl}benzoic acid
N-[(1-methylpiperidin-3-yl)methyl]-N-(2-phenylethyl)quinoxaline-5-carboxamide
2-(dimethylamino)-1-[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]-2-(2-methylphenyl)ethan-1-one
2-{2-[(2,4-dimethyl-1,4-diazepan-1-yl)methyl]-4-(pyridin-3-yl)phenoxy}acetic acid
6-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-methyl-1,3-benzoxazole
2-methyl-4-[methyl({[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl})amino]butan-2-ol
N-ethyl-6-fluoro-N-(propan-2-yl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline-4-carboxamide
2-(4-{[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]methyl}phenoxy)ethan-1-ol
3-[(3-{[(2R)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}phenyl)formamido]-N,N-dimethylpropanamide
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}-3-(1-methyl-1H-pyrazol-5-yl)propanamide
2-methoxy-4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}phenol
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(oxan-4-yl)ethyl]acetamide
1-(3,5-difluoropyridine-2-carbonyl)-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
6-cyano-N-methyl-N-[(4-phenoxyphenyl)methyl]pyridine-3-carboxamide
3-(1-methyl-1H-pyrrol-2-yl)-N-[(2-phenoxypyridin-3-yl)methyl]-1H-pyrazole-5-carboxamide
N-ethyl-5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidin-2-amine
1-methyl-N-[(3-propyl-1,2-oxazol-5-yl)methyl]-3-(thiophen-2-yl)-1H-pyrazole-5-carboxamide
3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1-methyl-1-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
1-(2,3-dihydro-1H-indene-5-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-{[4-cyclopentyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-2-methoxyphenol
4-(5-chloro-2-methoxyphenyl)-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
1-[({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]cyclohexan-1-ol
3-(4-propylphenyl)-5-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
1-cyclohexyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}-1H-imidazole
6-methyl-4-(pyridin-3-yl)-5-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,2,3,4-tetrahydropyrimidin-2-one
3-{1-[2-(2-methyl-1H-imidazol-1-yl)acetyl]piperidin-3-yl}benzoic acid
2-(2-propyl-1,3-thiazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-({cyclopropyl[(3-hydroxyphenyl)methyl]amino}methyl)-7-methyl-1,2-dihydroquinolin-2-one
2-[3-(1H-imidazol-1-yl)propyl]-9-(2-methyloxolane-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N3-tert-butyl-1-cyclohexyl-N5-[2-(1H-indol-3-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-cyclohexyl-4-{[1-(1H-imidazol-2-yl)ethyl]sulfamoyl}benzamide
3-(azetidine-1-carbonyl)-N-[3-(4-methylpiperazin-1-yl)propyl]benzene-1-sulfonamide
(3R,5S)-N3-(4-fluorophenyl)-N5-[2-(1H-indol-3-yl)ethyl]-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
(2E)-N-(2-{5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-fluorophenyl)-4H-1,2,4-triazol-3-yl}ethyl)-3-(thiophen-2-yl)prop-2-enamide
[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl][(1-methylpiperidin-4-yl)methyl](2-phenylethyl)amine
2-(1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)ethan-1-ol