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5-(methoxymethyl)-3-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1,2,4-oxadiazole
1-methyl-6-propyl-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[3-(3-chlorophenyl)phenyl]-1-[3-(methylsulfanyl)propanoyl]piperidine-4-carboxamide
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-[(5-propylfuran-2-yl)methyl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-methyl-4-{3-[4-(thian-4-yl)piperazine-1-carbonyl]phenyl}butan-2-ol
1-[2-(4-chlorophenyl)morpholin-4-yl]-3-(4-hydroxyphenyl)propan-1-one
(3R,4R)-1-cyclobutanecarbonyl-4-[(pyridin-3-ylmethyl)amino]pyrrolidin-3-ol
2-amino-2-methyl-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-one
(3S,4R)-1-(2,3-dihydroxybenzoyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-(2-methyl-1,3-benzothiazol-6-yl)-1-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]methyl}urea
6-(1,2-oxazolidin-2-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N-{2-[(2-methyl-1H-imidazol-1-yl)methyl]phenyl}-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
1-{3-[4-(4-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
N-cyclopentyl-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}-3-(2-oxopyrrolidin-1-yl)benzamide
6-[(1H-imidazol-2-ylmethyl)(methyl)amino]-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
3-[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazine-1-carbonyl]phenol
2-{[1-(1H-1,3-benzodiazol-2-yl)ethyl]amino}-N-(4-chloro-3-methoxyphenyl)acetamide
1-[(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
(3S,4R)-3-[(dimethylsulfamoyl)amino]-N-(4-methylphenyl)-4-(propan-2-yl)pyrrolidine-1-carboxamide
1-[3-(cyclopentyloxy)phenyl]-3-ethyl-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
3-[4-(dimethylamino)azepane-1-carbonyl]-1-ethyl-6-methyl-1,2-dihydropyridin-2-one
1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-methylurea
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylprop-2-en-1-yl)acetamide
N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]pyrimidin-4-amine
8-(3-aminopropanoyl)-2-[(3,4-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(1-ethyl-1H-imidazol-5-yl)methyl]-4-[(2,6,6-trimethylcyclohex-1-en-1-yl)methyl]-1H-1,2,3-triazole
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-1H-pyrazole-4-carbonyl)piperidine-4-carboxamide
8-(5-chloro-6-oxo-1,6-dihydropyridine-3-carbonyl)-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
1-tert-butyl-4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]pyrrolidin-2-one
2-(dimethylamino)-8-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
2-(4-chlorophenyl)-4-[3-(1H-pyrazol-4-yl)benzoyl]morpholine
methyl[2-methyl-3-(pyrrolidin-1-yl)propyl]{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
2-(1-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-4-yl)acetamide
1-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-(7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)pyridine-3-carboxamide
(1R,7S)-3-[(2,5-dimethylphenyl)methyl]-N-(1H-imidazol-2-ylmethyl)-N-methyl-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(thiophen-2-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{1-[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]piperidin-4-yl}methanesulfonamide
N-(3,4-dimethylphenyl)-1-(quinoxaline-5-carbonyl)piperidin-3-amine
4-cyano-N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-1H-pyrrole-2-carboxamide
2-(3-fluorophenyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}piperidine
2-ethyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]pyrazin-2-amine
1-(3-phenylpropyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepane
1-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]cyclobutan-1-amine
(3aR,6aR)-2-acetyl-5-[(4-phenyl-1,3-thiazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(2-hydroxypyridin-3-yl)-3-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)benzamide
1-methanesulfonyl-4-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]-1,4-diazepane