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(4aR,8aR)-7-(3-cyano-4,6-dimethylpyridin-2-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
1-(2H-1,3-benzodioxole-5-carbonyl)-4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidine
N-{[3-(difluoromethoxy)phenyl]methyl}-5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidin-2-amine
2,5-dioxo-6-pentyl-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-methyl-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-3-phenylpiperidine
(8aS)-2-(2-oxo-2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-(4-{[4-(benzyloxy)-3-methoxyphenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
6-ethyl-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
4-{[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
6-(methoxymethyl)-1-methyl-N-{2-[2-(propan-2-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
5-(2-fluorophenoxymethyl)-N-(2-hydroxyethyl)-N-methyl-1H-pyrazole-3-carboxamide
3-(azepane-1-carbonyl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]benzene-1-sulfonamide
N-[2-(dimethylsulfamoyl)ethyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
1-{[1-(4-methoxyphenyl)-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-5-yl]methyl}pyrrolidin-2-one
2-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-ethyl-1H-imidazole
4-hydroxy-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[1-(4-fluorophenyl)-2-hydroxyethyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
5-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
1-[bis(4-fluorophenyl)methyl]-4-(1-methylpyrrolidine-3-carbonyl)piperazine
5-(2-methoxyphenoxymethyl)-N-(3-methylbutyl)-1H-pyrazole-3-carboxamide
[1-({1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
N-(2-hydroxyethyl)-N-{[4-(methylsulfanyl)phenyl]methyl}-2-(pyridin-4-ylsulfanyl)acetamide
2-{[2-(pyridin-2-yl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
3-{2-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
(1R,5S,6S)-6-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}-3-azabicyclo[3.1.0]hexane
N-[(5-methylfuran-2-yl)methyl]-2-(pyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
5-ethyl-2,3-dimethyl-N-(oxan-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(pyridin-4-yl)propanamide
2-(1-cyclopentyl-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl)ethan-1-ol
N-(furan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-[(3S,4R)-1-[2-(4-fluorophenoxy)acetyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
2-({3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1-methyl-1H-indole
7-fluoro-4-{3-[(4-methylpiperazin-1-yl)methyl]piperidin-1-yl}quinazoline
(1R,5S,6S)-3-[(2-hydroxy-3,5-dimethylphenyl)methyl]-N-methyl-N-(pyrazin-2-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
4-methyl-5-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrimidine
1-[2-(4-fluorophenyl)pyrrolidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]but-3-enamide
(1S,5R)-3-cyclobutanecarbonyl-6-(3,4-difluorobenzoyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 4-[3-({[1-(4-chlorophenyl)cyclopropyl]formamido}methyl)piperidin-1-yl]-4-oxobutanoate
N-(1-hydroxybutan-2-yl)-3-methyl-1-propyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1H-pyrrol-1-yl)propan-1-one
N-butyl-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-4-oxo-4H-chromene-3-carboxamide
N-{[3-methyl-7-(9-methyl-9H-carbazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1,3-thiazole-5-carboxamide
ethyl 2-(1-{5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-1H-pyrazol-4-yl}-N-methylformamido)acetate
N-methyl-N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
N-(2-methoxyethyl)-4-(1-methyl-1H-indazol-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-5-methylthiophene-2-carboxamide
N2-(6-methoxypyrimidin-4-yl)-N1-(3-methylpyridin-2-yl)ethane-1,2-diamine