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N-[2-(3-methanesulfonamidopropyl)-4-methylphenyl]-3-methoxybenzamide
N-[2-methyl-1-oxo-1-(5-oxo-1,4-diazepan-1-yl)propan-2-yl]thiophene-2-carboxamide
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(2-phenoxyethyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
2-[3-({8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)phenoxy]acetamide
({4-ethyl-5-[1-(6-methyl-2-propylpyrimidin-4-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]propanamide
N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
1-methyl-4-{[2-(methylamino)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-6-yl]methyl}-1H-pyrrole-2-carbonitrile
N-[2-(furan-2-yl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-(piperidin-4-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}pyrimidin-4-amine
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(2-methylpropyl)piperidine-4-carboxamide
propan-2-yl 2-chloro-5-({methyl[3-(1H-pyrazol-1-yl)propyl]carbamoyl}amino)benzoate
1-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(piperidin-1-yl)propan-2-ol
6-amino-N-[(5-ethylpyridin-2-yl)methyl]-N-methylpyridine-2-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-2,8-dimethylquinoline-4-carboxamide
ethyl({[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl})[(1-methylpyrrolidin-3-yl)methyl]amine
[3-({1-[1-(4-methoxyphenyl)piperidin-4-yl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-3-phenyl-1,2-oxazole-5-carboxamide
(3-phenylpropyl)({[6-(pyrrolidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
N-methyl-2-(4-{1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)acetamide
1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-4-(1H-imidazol-2-yl)piperidine
2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-1-[4-(pyridin-3-yl)piperazin-1-yl]ethan-1-one
(3aR,6aR)-2-(1H-imidazol-4-ylmethyl)-5-(quinolin-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-cyclopentyl-1-methyl-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
8-(2,3-dihydro-1H-inden-2-yl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
6-methyl-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propylimidazo[2,1-b][1,3]thiazole-5-carboxamide
N-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenyl-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
2,6-dimethyl-3-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,4-dihydropyridin-4-one
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[1-(3-methylphenyl)piperidin-4-yl]pyrrolidin-3-yl]methanol
N-(4,6-dimethyl-2-oxo-1,2-dihydropyridin-1-yl)-3-(2-methoxyphenyl)propanamide
N-(3-hydroxypropyl)-2,6-dimethyl-N-[(4-methylphenyl)methyl]pyridine-4-carboxamide
7-methyl-2-[3-(2-methylphenyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
6-(4-methylpiperazin-1-yl)-N4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}pyrimidine-2,4-diamine
5-(1H-imidazol-1-ylmethyl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyridin-2-amine
1-{1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-1H-pyrazole-4-carbonyl}-4-methyl-1,4-diazepane
6-methoxy-3-{[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
5-(1-methyl-4-phenyl-1H-imidazol-5-yl)isoquinoline
N-(butan-2-yl)-N-cyclopentylimidazo[1,2-a]pyridine-6-carboxamide
[(3-chloro-4,5-diethoxyphenyl)methyl](methyl)[1-(pyridin-2-yl)ethyl]amine
ethyl 5-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-1-(2-methoxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-benzyl-4-(2,4-dimethylquinoline-7-carbonyl)piperazin-2-one
2-(dimethylamino)-4-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]pyrimidine-5-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-2-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
3-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
N-[2-ethyl-4-(1-methyl-1H-pyrazol-4-yl)phenyl]acetamide
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-[(2-fluorophenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(furan-2-amido)-N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
4-(4-{[1-(1H-indol-1-yl)propan-2-yl]amino}piperidin-1-yl)-N,N-dimethylbenzamide
4-(4-methylphenoxy)-N-[3-(oxolan-3-yl)propyl]piperidine-4-carboxamide