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1-(1-methyl-1H-pyrazole-5-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
2-amino-4-cyclopropyl-6-(3,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
4-[3-(3,3-diethylpyrrolidine-1-carbonyl)phenyl]-2-methylbutan-2-ol
(1R,5R)-N,N-dimethyl-6-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
3,5-dimethyl-N-[3-(1H-1,2,3-triazol-1-yl)propyl]-1H-indole-2-carboxamide
(dicyclopropylmethyl)({[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
3-[(dimethylamino)methyl]-1-(4-methyl-1H-imidazole-5-carbonyl)piperidin-3-ol
1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-8-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-ethyl-3-(1-{4-methyl-3-oxo-1H,2H,3H-pyrazolo[3,4-b]pyridine-6-carbonyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-ethyl-N-(2-hydroxyethyl)-5-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,3-thiazole
2-(4-chloro-2-methylphenoxy)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]propan-1-one
4-{2-[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}morpholine
N-(2-methoxyethyl)-2-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
N,3,5,7-tetramethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-indole-2-carboxamide
(1S,5R)-6-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{3-[3-(3-ethylphenoxy)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
3-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)-7-methoxy-1,2-dihydroquinolin-2-one
5-[2-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)-2-oxoethyl]imidazolidine-2,4-dione
N,1-dimethyl-6-oxo-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1,6-dihydropyridazine-3-carboxamide
(3aR,6aR)-2-(4-tert-butylbenzoyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}-6-(propan-2-yloxy)pyrimidin-2-amine
2-[2-(dimethylamino)ethyl]-8-(4-methyl-1H-imidazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
8-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-butyl-4-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-1-methylpiperazin-2-one
1-[(4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}phenyl)methyl]-1H-pyrazole
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1,6-dimethyl-1,4-dihydroquinolin-4-one
1-[1-(2,3-difluoro-4-methoxybenzoyl)piperidin-4-yl]piperidin-3-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine
5-(morpholin-4-yl)-2-(oxolan-2-ylmethyl)-2,3-dihydropyridazin-3-one
3-(2-{1,3-dimethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1H-pyrrol-1-yl)pyridine
8-{[3-(3-chlorobenzoyl)piperidin-1-yl]sulfonyl}quinoline
3-{[2-(2-aminoethyl)quinazolin-4-yl][(4-fluorophenyl)methyl]amino}propan-1-ol
2-methoxy-3-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-2-[methyl(pyridin-3-ylmethyl)amino]acetamide
4-amino-5-[4-(dimethylamino)phenyl]-2-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
1-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-3-(1-methylpiperidin-2-yl)propan-1-one
1-[4-hydroxy-4-(2-methylquinolin-6-yl)piperidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
3-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-1-methyl-1-[(3-methylpyridin-4-yl)methyl]urea
N-[(3,4-dimethoxyphenyl)methyl]-2-ethyl-N-(pyridin-4-ylmethyl)butanamide
2-hydroxy-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-4-methylpentan-1-one
2-{[(4aS,8aR)-1-(4-hydroxybutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]methyl}benzonitrile
5-[4-(5-methylpyrimidin-2-yl)phenyl]-1,2-dihydropyridin-2-one
2-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazole
3-{1-[5-(2-chlorophenyl)furan-2-carbonyl]pyrrolidin-2-yl}pyridine
3-(dimethyl-1,2-oxazol-4-yl)-1-[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]propan-1-one
N4-{[1-(ethoxymethyl)cyclobutyl]methyl}-5-ethylpyrimidine-2,4-diamine