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2-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-8-methyl-2,8-diazaspiro[5.5]undecane
(3S)-N-tert-butyl-2-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-(3-{1-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
N,N-dimethyl-2-[(1S,5R)-3-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
[(6-ethoxyquinolin-2-yl)methyl](methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
(2S)-1-[2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carbonyl]pyrrolidine-2-carboxamide
4,5-dimethyl-3-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-2,3-dihydro-1,3-oxazol-2-one
2-(4-methoxy-3-{[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}phenyl)acetic acid
2-[4-(2-methyl-4-phenylpyridine-3-carbonyl)piperazin-1-yl]pyrimidine
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{[3-(5-methylfuran-2-yl)phenyl]methyl}-2-(pyridin-3-yl)morpholine
2-(3-methoxyphenyl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidine
1-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]imidazolidine-2,4-dione
3-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-(2-phenylethyl)urea
9-[(2-phenyl-1,3-oxazol-4-yl)methyl]-6-oxa-9-azaspiro[4.5]decane
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-(6-phenoxypyridin-3-yl)piperidine-4-carboxamide
3-methyl-4-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-4H,5H,6H,7H-[1,2]thiazolo[5,4-b]pyridin-6-one
(3S,4S)-1-(2-methoxy-2-methylpropanoyl)-4-propylpyrrolidine-3-carboxylic acid
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-N-(furan-2-ylmethyl)pyridine-2-carboxamide
(2R,4S)-1-[(2-chloro-3,4-dimethoxyphenyl)methyl]-4-hydroxypiperidine-2-carboxylic acid
(2S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(dimethylamino)pyrrolidine-2-carboxylic acid
(3S,5R)-N3-cyclopentyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
1-[(1S,5R)-6-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
3-chloro-4-fluoro-N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]benzene-1-sulfonamide
13-(3,4-dimethylphenyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-6-methylpyridine
2-{4-[(3S)-3-hydroxy-3-phenylpropyl]-2-oxopiperazin-1-yl}benzonitrile
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(2-methyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methanol
N-(6-phenoxypyridin-3-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidine-4-carboxamide
1-(4-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}piperidin-1-yl)-3-methylbutan-1-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
3-(methanesulfonylmethyl)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]piperidine
6-(cyclohex-3-en-1-ylmethyl)-N-[(1-phenylcyclopentyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1-carbamoylcyclopentyl)-1,3-oxazole-4-carboxamide
N,N-dimethyl-2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
1-[(butan-2-yl)carbamoyl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-methyl-1-[3-(2-phenylethyl)-1H-1,2,4-triazole-5-carbonyl]-2,3-dihydro-1H-indole
2-(2-chlorophenyl)-2-{[3-(1H-pyrazol-1-ylmethyl)phenyl]formamido}acetic acid
N,5,7-trimethyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
(2R,3R)-1'-(4-amino-5-fluoropyrimidin-2-yl)-3-(morpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N-[3-(cyclohexyloxy)propyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
4-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxymethyl]-2-(furan-2-yl)-5-methyl-1,3-oxazole
N-methyl-2-phenyl-N-[1-(pyridin-2-yl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
2-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}-5,8-dimethyl-1,4-dihydroquinolin-4-one
(2R)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
(3R,4R)-1-[2-methyl-2-(morpholin-4-ylmethyl)propyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
2-(5-methyl-1H-pyrazol-1-yl)-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
(4aR,7aS)-4-(4-chlorobenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-(furan-2-ylmethyl)-4-{4-[(methylamino)methyl]-1H-1,2,3-triazol-1-yl}piperidine-1-carboxamide