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1-(1-ethylpiperidin-4-yl)-3-(6-methoxynaphthalene-2-carbonyl)piperidine
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-(2-oxo-4-phenylpyrrolidin-1-yl)acetamide
2-(3-butyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
N-[1-(7-{[4-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]methanesulfonamide
2-amino-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-phenylpyrimidine-5-carboxamide
2-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[2-(pyrazin-2-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-1-cyclopentyl-5-oxopyrrolidine-3-carboxamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidin-2-one
1-[2-(1,3-benzoxazol-2-yl)ethyl]-3-[1-(propan-2-yl)-1H-pyrazol-4-yl]urea
1-{2-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
3-[2-amino-4-methyl-6-({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)pyrimidin-5-yl]propanoic acid
2-(2-{1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-4-methylpyrimidine-5-carboxamide
3-(piperidine-1-carbonyl)-1-propyl-N-[2-(pyridin-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl 3-[(4-fluorophenyl)methyl]-1-(8-fluoroquinoline-2-carbonyl)piperidine-3-carboxylate
2-chloro-5-[1-(1,4-dioxan-2-ylmethyl)-1H-1,2,3-triazol-4-yl]pyridine
1-[(4aR,8aR)-7-(2-amino-5-ethylpyrimidin-4-yl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
2-amino-4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]-6-(trimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
N-[1-(cyclohex-1-en-1-yl)ethyl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
1-ethyl-5-[(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
7-(1,3-benzothiazol-2-yl)-4-(quinolin-4-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
1-{[2-(3-chlorophenyl)-8-methylquinolin-3-yl]methyl}-1,4-diazepan-5-one
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
6-[1-(4,6-dimethoxypyrimidin-2-yl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-[(4-acetylmorpholin-2-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
3-[1-(1-methylpiperidin-4-yl)-5-(pyridin-3-ylmethyl)-1H-1,2,4-triazol-3-yl]pyridine
1-{2-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]phenyl}-1,3-diazinane-2,4-dione
4-methyl-2-(propan-2-yl)-5-[3-(pyrrolidin-1-yl)piperidine-1-carbonyl]pyrimidine
2-methyl-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
ethyl 4-{1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperazine-1-carboxylate
2-(3-{[7-methyl-2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenoxy)ethan-1-ol
1-methyl-4-{1-[1-(4-methylpyridin-2-yl)-3-pentyl-1H-1,2,4-triazol-5-yl]ethyl}piperazine
N-[(1-ethylpiperidin-3-yl)methyl]-1,5-dimethyl-1H-indazole-3-carboxamide
N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-3-(1H-1,2,4-triazol-3-yl)benzamide
N-methyl-N-[(2-methyl-1H-1,3-benzodiazol-5-yl)methyl]oxan-4-amine
4-(1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)pyrimidine
3-{[2-(5-tert-butyl-1H-pyrazol-3-yl)-1H-imidazol-1-yl]methyl}-5-(furan-2-yl)-1,2-oxazole
{4-[(2-chlorophenyl)methyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}methanol
1-amino-N-butyl-N-[(2-methylphenyl)methyl]cyclopropane-1-carboxamide
1-(propan-2-yl)-N-[1-(pyrazin-2-yl)piperidin-4-yl]-1H-pyrazole-4-carboxamide
2-(2-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}phenoxy)acetic acid
4-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-2-amine
4-(3,4-dichlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-(furan-2-ylmethyl)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}piperidine-3-carboxamide
6-[1-(1,5-dimethyl-1H-indole-2-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-ol
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
N-({1-[(2-methylpyrimidin-5-yl)methyl]pyrrolidin-3-yl}methyl)pyridine-4-carboxamide
4-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2-(trifluoromethyl)morpholine