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3-(2-methylphenyl)-5-{thieno[3,2-d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
2-{4-[2-(1-methyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]phenyl}-1H-1,3-benzodiazole
5-[1-(5-acetylthiophene-3-carbonyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
N-[(3R,4R)-3-hydroxy-1-[3-(methylsulfanyl)propyl]piperidin-4-yl]pyrazine-2-carboxamide
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(pyridin-2-yl)propanamide
2-(2,4-dioxoimidazolidin-1-yl)-N-[3-(4-methoxyphenoxy)propyl]-N-methylacetamide
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-hydroxyethan-1-one
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]benzamide
(3R,4R)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
2-({5-propylpyrazolo[1,5-a]pyrimidin-7-yl}amino)hexanamide
1-ethyl-4-{4-[(4-fluorophenyl)methyl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-(3-fluorophenoxymethyl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,3-oxazole-4-carboxamide
3,4,4-trimethyl-1-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-3-ol
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(2-hydroxyphenyl)ethan-1-one
1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-4-(2,2,2-trifluoroethyl)piperazine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2,3-dihydro-1,4-benzodioxine-6-carboxamide
4-(2-{4-[3-(1H-imidazol-2-yl)benzoyl]piperazin-1-yl}ethyl)morpholine
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-2-(thiophen-3-yl)acetamide
(3R,4S)-4-phenyl-1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]pyrrolidin-3-amine
6-[(3,5-dimethoxyphenyl)methyl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
9-(3-phenoxypropyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-methyl-8-[(6-phenoxypyridin-3-yl)methyl]-2,8-diazaspiro[4.5]decane
N-(2-{1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1,2,3,6-tetrahydropyridin-4-yl}ethyl)acetamide
4-(1H-1,2,3-benzotriazole-5-carbonyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
(1S,3R)-3-amino-N-(2-methanesulfonamido-5-methoxyphenyl)cyclopentane-1-carboxamide
2-(2-methoxy-5-{[(1R,6S)-9-methyl-3,9-diazabicyclo[4.2.1]nonan-3-yl]methyl}phenoxy)acetic acid
N-cyclopentyl-3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-3-ylmethyl)piperidin-3-yl]propanamide
3-[(cyclohex-1-en-1-ylmethyl)sulfamoyl]-N-(oxolan-2-ylmethyl)benzamide
[2-(3,4-dimethoxyphenyl)ethyl](methyl){[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(piperazin-1-yl)-2-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-(4-methoxybutyl)-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
[(3,5-difluorophenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
3-(4-methoxy-2-methylbenzoyl)-1-phenylmethanesulfonylpiperidine
N-[2-(1H-indol-1-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
(4S)-3-{2-[4-(furan-3-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-4-(propan-2-yl)-1,3-oxazolidin-2-one
2-(adamantan-1-yl)-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
2-{[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]methyl}benzonitrile
4-[(2,6-difluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]piperidine
5-cyclopropyl-N-[2-(4-sulfamoylphenyl)ethyl]-1,3-oxazole-4-carboxamide
2-(acetamidomethyl)-N-(2,4,6-trimethylpyridin-3-yl)-1-oxa-8-azaspiro[4.5]decane-8-carboxamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(1S,2R)-2-[(2,3-dihydro-1H-inden-2-yl)amino]cyclobutyl]-2H-1,3-benzodioxole-5-carboxamide
2-[4-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-2-oxopiperazin-1-yl]benzonitrile
1-[(5-ethylfuran-2-yl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-cyclohexyl-1-(pyridin-3-ylmethyl)-3-(3-sulfamoylphenyl)urea
5-chloro-2-[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]-1H-1,3-benzodiazole
3-(2,3-dihydro-1H-inden-2-yl)-1-(3-methanesulfonamido-4-methoxyphenyl)-3-methylurea
2-(2H-1,3-benzodioxole-5-carbonyl)-7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane