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N,1-dimethyl-N-[(3-methyl-1H-indol-2-yl)methyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-cyclobutyl-2-(4-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}morpholin-3-yl)acetamide
1-[4-(6,7-dimethoxy-1-methyl-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)thiophen-2-yl]ethan-1-one
3-(4-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
(1S,5R)-6-(cyclopropylmethyl)-3-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{2-[(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}piperidin-4-yl)formamido]ethyl}acetamide
5-{[methyl({[3-(2-{4-[2-(trifluoromethoxy)benzenesulfonyl]piperazin-1-yl}ethoxy)phenyl]methyl})amino]methyl}pyrrolidin-2-one
3-(1-methyl-1H-pyrazol-4-yl)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}propanamide
2-(3-hydroxypropyl)-9-(1H-indol-5-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-benzyl-3-[(2-methyl-1,3-thiazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-cyclopropylpropan-1-one
2-[4-(1H-pyrazol-5-yl)phenyl]benzamide
1-(4-methylpentanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-[(4,6-dimethylquinolin-2-yl)sulfanyl]propan-1-one
3-[(1-methanesulfonylpiperidin-3-yl)methyl]-1-[4-(1H-1,2,4-triazol-1-yl)phenyl]urea
2-[(2-chlorophenyl)methyl]-4-(4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]hexane-1,5-dione
N-[2-(2-fluorophenyl)-1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylthiophene-3-carboxamide
4-(4-methylphenoxy)-1-(pyridin-4-ylmethyl)piperidine-4-carboxylic acid
N-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
1-{2-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}ethan-1-one
4-[(5-methylfuran-2-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridine-2-carbonitrile
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
3-(1H-pyrazol-3-yl)-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidine
2-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-(2-ethoxyethyl)-N-(1H-imidazol-2-ylmethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-ethyl-8-[(5-fluoro-3-methyl-1H-indol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-{2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-1-(2-phenylethyl)piperazin-2-one
ethyl 1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-imidazole-2-carboxylate
(4aR,7aS)-1-acetyl-4-(3-hydroxy-2-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclobutanecarboxamide
7-[(4-fluorophenyl)methyl]-2-(furan-2-carbonyl)-2,7-diazaspiro[4.5]decane
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-1-[4-(2-methylphenoxy)piperidin-1-yl]propan-1-one
6-chloro-3-fluoro-N-methyl-N-[1-(pyridin-3-yl)pentyl]imidazo[1,2-a]pyridine-2-carboxamide
5-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-2-methyl-1H-1,3-benzodiazole
2-amino-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-6-(2-methylpropyl)pyrimidine-4-carboxamide
5-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-cyclopentyl-4-(6-ethoxypyridazin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{1-[(4-ethoxyphenyl)methyl]-4-(5-ethyl-2-methylpyrimidin-4-yl)piperazin-2-yl}ethan-1-ol
2-{9-[(2-ethoxyphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
1-cyclohexyl-1-(2-hydroxyethyl)-3-[3-(2-methoxyphenyl)phenyl]urea
8-[3-(methylsulfanyl)propanoyl]-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N3-(1-benzylpiperidin-4-yl)-N5-ethyl-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-({7-[(9-ethyl-9H-carbazol-3-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)propane-2-sulfonamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperazine
2-[4-(4-cyanophenyl)-1H-pyrazol-1-yl]-N-(1-phenyl-1H-pyrazol-5-yl)acetamide
N-[2-(4-fluorophenyl)ethyl]-2-[(oxan-2-ylmethyl)amino]acetamide
(3R,4S)-4-{[(3-chloro-4-fluorophenyl)methyl](methyl)amino}oxolan-3-ol
(5S)-5-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]pyrrolidin-2-one