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(1r,4r)-4-methyl-N-(2-{4-[(1-methyl-1H-pyrazol-4-yl)methyl]morpholin-2-yl}ethyl)cyclohexane-1-carboxamide
2-{1-cyclohexyl-4-[(3,4-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-[2-(aminomethyl)morpholin-4-yl]-N-cyclopentyl-2-oxoacetamide
4-{5-benzoyl-1-benzyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}morpholine
(2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-8-methylquinolin-3-yl)methanol
8-[2-(4-chlorophenyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperazine
N-(1-{1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
1-(furan-2-ylmethyl)-5-(oxolan-3-yl)-4-phenyl-1H-imidazole
4-(3,3-difluoropiperidine-1-carbonyl)-7,8-dimethyl-2-(2-methylpyrimidin-5-yl)quinoline
3-(4-phenoxybenzoyl)-1-(1,2,5-thiadiazole-3-carbonyl)piperidine
N-(3-chloro-4-methylphenyl)-N'-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}propanediamide
4-benzyl-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-2-one
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
3-{1-[(8-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
(3R,4R)-4-cyclopropyl-1-{[2-fluoro-5-(trifluoromethyl)phenyl]methyl}-3-methylpiperidin-4-ol
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}morpholine-2-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]benzamide
4-{[({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]methyl}-2-methoxyphenol
1-(2,3-dihydro-1H-inden-2-yl)-4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazine
1-[(4-fluorophenyl)methyl]-5-{furo[3,2-c]pyridin-4-yl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole
3-{1-[4-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)piperidin-1-yl]-1-oxopropan-2-yl}-3,4-dihydroquinazolin-4-one
8-(2H-1,3-benzodioxol-5-yl)quinoline
N-[2-(benzylsulfanyl)ethyl]-1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[3-(hydroxymethyl)piperidin-1-yl]-N-propylpyridine-3-carboxamide
5-[2-({5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
7,7-dimethyl-2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(2-oxo-5,5-diphenylpiperidin-1-yl)-N-(propan-2-yl)acetamide
4-methoxy-N-({1-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-3-yl}methyl)benzene-1-sulfonamide
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(4-methylphenyl)quinoline-4-carboxamide
N-[(1S,2R)-2-[(1-acetylpiperidin-4-yl)amino]cyclobutyl]pyridine-3-sulfonamide
ethyl 1-(1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carbonyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
1-(2-{4-[(dimethylamino)methyl]phenyl}piperidin-1-yl)-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
3-methyl-N-[2-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
N-benzyl-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
6-[2-amino-7-methyl-4-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-2,2-dimethyl-3,4-dihydro-2H-pyran-4-one
N-[(4-methylphenyl)methyl]-2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carboxamide
N-[2-(benzyloxy)phenyl]-6-[(dimethylamino)methyl]-1,4-oxazepane-4-carboxamide
3-{3-[(3,4-difluorophenyl)amino]piperidine-1-carbonyl}-N-methylpyridin-2-amine
6-methyl-2-oxo-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-4-carboxamide
1-({1-[1-(pentan-2-yl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)azepane
3-{2-[2-(furan-3-yl)-1H-imidazol-1-yl]ethyl}-2-methyl-1H-indole-5-carbonitrile
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methoxyethyl)acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{[4-(4-hydroxy-2-methylpyrimidine-5-carbonyl)piperazin-1-yl]methyl}benzonitrile
5,5-dimethyl-3-{2-oxo-2-[3-oxo-4-(2-phenylethyl)piperazin-1-yl]ethyl}-1,3-oxazolidine-2,4-dione
N-[3-(3,5-dimethylphenoxy)propyl]-2-ethyl-N-methylpyrimidine-5-carboxamide
methyl 3-{[1-(1-benzylpiperidin-4-yl)piperidin-3-yl]formamido}propanoate