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1-benzyl-5-(furan-3-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
2-(2-chloro-4-fluorophenoxymethyl)-N-methyl-N-(pyrazin-2-ylmethyl)-1,3-oxazole-4-carboxamide
ethyl 5-{[bis(2-hydroxyethyl)amino]methyl}-1-(7-chloroquinolin-4-yl)-1H-pyrazole-4-carboxylate
(2R,3R)-3-{methyl[(3-methyl-1H-indol-2-yl)methyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
[(4aS,8aR)-6-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
N-cyclopropyl-1,3-dimethyl-N-(pyridin-3-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
8-{imidazo[1,2-a]pyrimidine-2-carbonyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
3-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]urea
methyl 3-[(2S)-2-carbamoylpyrrolidine-1-carbonyl]-5-(cyclobutylmethoxy)benzoate
2-(1H-pyrazol-1-yl)-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)acetamide
9-(6-methyl-2-propylpyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-1-(8-fluoro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
2-fluoro-N-{4-[4-({[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}amino)piperidin-1-yl]phenyl}benzamide
methyl 2-[2-(3-hydroxy-3-phenylpyrrolidin-1-yl)acetamido]-4-methyl-1,3-thiazole-5-carboxylate
1-[(4-hydroxyphenyl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
(3aS,6aS)-2-[5-(1H-imidazol-2-yl)thiophene-2-carbonyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3-{3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}phenyl)-1H-imidazole
6-{4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}-9H-purine
2-cyclopentyl-N-{3-[4-(morpholin-4-ylmethyl)phenoxy]propyl}acetamide
ethyl 4-{3-oxo-2,8-diazaspiro[4.5]decan-8-yl}piperidine-1-carboxylate
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(1H-1,2,4-triazol-3-yl)benzamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(3-phenylbenzoyl)pyrrolidin-3-yl]methanol
2-{9-[(3-cyanophenyl)carbamoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
N-(1-methyl-1H-pyrazol-5-yl)-4-{[(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]methyl}benzamide
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-(2-methylphenyl)pyrrolidin-3-ol
4-{5-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
3-[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]quinoline
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-methylpiperazin-2-yl]ethan-1-ol
3-[(3R,4S)-1-(2-chloro-5-fluorobenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-[(5-methoxy-1H-indol-2-yl)methyl]-3-methyl-1H-pyrazole-5-carboxamide
8-[2-(2,3-dimethoxyphenyl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
(1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-3-[(2-methylphenyl)methyl]piperidin-3-yl)methanol
2-(3-hydroxypiperidin-1-yl)-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylacetamide
2-[4-(1-methoxyethyl)phenyl]-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
4-fluoro-3-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]benzene-1-sulfonamide
3-[2-(naphthalen-1-yl)ethyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[4-(hydroxymethyl)benzoyl]-3-methyl-1-[(4-methylphenyl)methyl]piperazin-2-one
N-(1-benzyl-5-oxopyrrolidin-3-yl)-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-{[(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
4-[1-(methoxymethyl)cyclopropanecarbonyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
1-[(3-fluorophenyl)methyl]-4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine
N-[(3R,4S)-1-(2-hydroxyethyl)-4-propylpyrrolidin-3-yl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-(1H-pyrazol-1-ylmethyl)benzamide
4-hydroxy-N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-(thian-4-yl)pyrimidine-5-carboxamide
2-[2-(morpholine-4-carbonyl)pyridin-4-yl]-2,3-dihydro-1H-isoindole
2-{1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-2-yl}-5-fluoro-1H-1,3-benzodiazole
2-amino-4-(1-methyl-1H-pyrazol-4-yl)-6-[2-(propan-2-yloxy)phenyl]pyridine-3-carbonitrile
4-chloro-N,N-dimethyl-5-{1-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-1H-imidazol-2-yl}-1,3-thiazol-2-amine