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N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
1-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(4H-1,2,4-triazol-4-yl)ethan-1-one
3-{2-oxo-2-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)pyrrolidin-1-yl]ethyl}-3,4-dihydroquinazolin-4-one
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
2-(3-fluorophenyl)-N-(1-methyl-1H-pyrazol-5-yl)azepane-1-carboxamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-[4-(thiophen-2-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]propan-1-one
[(3R,4R)-1-(3-chlorothiophene-2-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
{1-[4-(methylsulfanyl)benzoyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
(3-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)methanamine
N-(1-ethyl-5-oxopyrrolidin-3-yl)-7-fluoro-2-(1-methyl-1H-pyrazol-4-yl)quinoline-4-carboxamide
N-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-2-(2-oxoazonan-1-yl)acetamide
methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl][(2,6,8-trimethylquinolin-4-yl)methyl]amine
N-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-4,4-difluoropiperidine-1-carboxamide
(1S,5R)-6-[(4-chloro-3-fluorophenyl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]pyrazolo[1,5-a]pyridine-7-carboxamide
4-(2-amino-5-ethyl-6-methylpyrimidin-4-yl)-1-(3-methoxyphenyl)piperazin-2-one
5-fluoro-N4,N4-dimethyl-N2-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]pyrimidine-2,4-diamine
3-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]benzonitrile
1-cyclohexyl-4-[1-(propan-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1H-1,2,3-triazole
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-3-[5-(phenoxymethyl)-1,3,4-oxadiazol-2-yl]propanamide
({6-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyrazin-2-yl}methyl)dimethylamine
N4-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]pyrimidine-4,6-diamine
5-ethyl-2-methyl-N-[1-(4-methylbenzoyl)piperidin-4-yl]pyrimidin-4-amine
N,1,3-trimethyl-N-(3-methylbutan-2-yl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
7-(3-hydroxy-2-methylbenzoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl]formamido}-N-(1,3-thiazol-2-yl)acetamide
N-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3,4-dichlorobenzamide
2-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-8-(trifluoromethyl)-1,2,3,4-tetrahydroisoquinoline
1-(4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}phenyl)-1H-1,2,4-triazole
N-[2-(3-phenylpyrrolidin-1-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
N'1-[(3R,4S)-4-cyclopropyl-1-[(3-fluoro-5-methylphenyl)methyl]pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
2-(ethylamino)-N-{2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl}pyrimidine-5-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]benzamide
1-[(3-methylpyridin-2-yl)methyl]-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazine
5-[1-(5-chloro-2-methoxyphenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]pyrimidine
1-methyl-4-[1-(1-{[2-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)ethyl]piperazine
methyl (2S,4R)-4-hydroxy-1-{[(5-propyl-1,3,4-thiadiazol-2-yl)carbamoyl]methyl}pyrrolidine-2-carboxylate
3-(4-hydroxyphenyl)-N-[3-(morpholin-4-yl)propyl]-2-phenylpropanamide
{5-[(1R,5R)-3-azabicyclo[3.3.1]nonane-3-carbonyl]furan-2-yl}methanol
4-{[3-(oxan-4-yl)-7-{1H-pyrrolo[2,3-b]pyridin-6-yl}-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazin-5-yl]methyl}-1H-imidazole
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-{2-[1-(5-cyanopyridin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
2-methyl-8-(3-methylfuran-2-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-{2-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl}phenol
5,6-dimethyl-2-[3-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
N-ethyl-4-(2,3,4-trimethoxyphenyl)benzamide
5-{2-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
5-(2,4-difluorophenoxymethyl)-3-[3-(2-methylpropyl)pyrrolidine-1-carbonyl]-1,2-oxazole
N-[2-(7-methyl-1H-indol-3-yl)ethyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide