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N-cyclohexyl-1-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-3-carboxamide
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(2-amino-1,3-thiazol-4-yl)propan-1-one
6-(difluoromethyl)-2-(2-{[ethyl(pentan-2-yl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
3-{2-[4-(4-methylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
ethyl({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})[2-(1H-pyrazol-1-yl)ethyl]amine
N-({1-[(2-ethylphenyl)methyl]pyrrolidin-3-yl}methyl)propane-2-sulfonamide
4-[(3,5-dimethylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
3-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-N-[(4-methylphenyl)methyl]propanamide
4-{[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
ethyl 6-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-ylmethyl]pyrazolo[1,5-a]pyrimidine-3-carboxylate
6-({4-[1-(2-hydroxybutyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)-2-methylpyrimidin-4-ol
4,4-difluoro-N-[4-(4-methyl-4H-1,2,4-triazol-3-yl)phenyl]piperidine-1-carboxamide
[1-(1-benzothiophen-2-ylmethyl)-3-[(2,4-difluorophenyl)methyl]piperidin-3-yl]methanol
7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-2-(dimethylamino)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-({3-[(1S,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]-1,2-oxazol-5-yl}methyl)-2-methyl-1H-1,3-benzodiazole
4-hydroxy-2-(1H-1,2,4-triazol-1-ylmethyl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]pyrimidine-5-carboxamide
(2E)-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-3-(thiophen-2-yl)prop-2-enamide
N-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-N-{[4-(methylsulfanyl)phenyl]methyl}cyclopropanamine
4-{5-[1-(1H-indazol-6-yl)-1H-imidazol-2-yl]thiophen-2-yl}-2-methylbut-3-yn-2-ol
4-{[2-(3-methoxyphenyl)piperidin-1-yl]methyl}-2,1,3-benzoxadiazole
methyl (2S)-1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]pyrrolidine-2-carboxylate
N-(1-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}pyrrolidin-3-yl)acetamide
4-[2-(pyridin-3-yl)-1H-imidazol-1-yl]thiophene-2-carboxamide
1-[(1-{6-[(cyclohexylmethyl)amino]pyridine-3-carbonyl}piperidin-4-yl)methyl]pyrrolidin-2-one
(R)-[1-(2-methoxyphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl](phenyl)methanol
methyl 1-[(3R,5S)-1-[(2-hydroxyphenyl)methyl]-5-({[3-(trifluoromethyl)phenyl]methyl}carbamoyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
9-[2-(methylamino)pyridine-4-carbonyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
7-(cyclohexylmethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-ethyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
1-{[3-(benzyloxy)phenyl]methyl}-4-methyl-1,4-diazepan-5-one
1-(azocan-1-yl)-3-[4-({[3-(dimethylamino)propyl](methyl)amino}methyl)-2-methoxyphenoxy]propan-2-ol
1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(furan-2-yl)ethane-1,2-dione
1-[3-(5-methyl-1,2-oxazol-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
5-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-(5-{[4-(pyridin-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}furan-2-yl)benzonitrile
8-(3-aminopropanoyl)-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-4-(piperidin-1-yl)benzamide
1-[(4-chlorophenyl)methyl]-4-(pyrrolidin-3-ylmethyl)piperazine
5-(2H-1,3-benzodioxol-4-ylmethyl)-8-methoxy-2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N,N-dimethyl-4-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazine-1-sulfonamide
4-{5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
2-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1,2-oxazinane
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-1-methylpiperidine-4-carboxamide
N-{1-[1-(6-aminopyrimidin-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
4-(furan-2-ylmethyl)-2-[(3-methoxyphenyl)methyl]morpholine
3-(4-hydroxyphenyl)-2-phenyl-N-(pyridin-2-ylmethyl)propanamide
(2S,4S)-N-ethyl-4-[2-(morpholin-4-yl)acetamido]-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
3-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1,9-dioxaspiro[5.5]undecan-4-amine