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{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)methylamine
2-{[(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)amino]methyl}-6-fluoroquinolin-4-ol
3-{1-[5-(morpholin-4-yl)pentyl]-1H-imidazol-2-yl}benzonitrile
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(4-fluorophenyl)-2-hydroxyethan-1-one
5-chloro-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)pyridine-3-carboxamide
1-({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)-1,4-diazepan-5-one
N-(1-ethyl-5-oxopyrrolidin-3-yl)-1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazole-5-carboxamide
1-(4-{[(5-methylfuran-2-yl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2-(4-{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
(3S,4S)-1-(6-methoxypyrimidin-4-yl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
2-amino-4-[5-(2-methylpropyl)thiophen-2-yl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-ethyl-2-[2-oxo-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]acetamide
1-(2-{[(1-phenylcyclopropyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
4-(5-phenylthiophen-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
1-[2-(3-fluorophenyl)piperidin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
1-(3-cyano-4-methoxyphenyl)-3-[3-(propan-2-yloxy)propyl]urea
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-(3-chloro-4-fluorophenoxy)ethan-1-one
N-(2-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)acetamide
1-{2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]ethyl}pyrrolidin-2-one
2-methyl-1-{2-oxo-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]ethyl}-1H-indole-3-carbonitrile
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]propanamide
9-hydroxy-N-methyl-4-oxo-N-[1-(pyridin-3-yl)pentyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
(1R,3S,5S)-8-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octane
[1-(2,6-dimethylphenoxy)propan-2-yl]({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3,5-dimethyl-1H-1,2,4-triazole
3-{[1-(ethoxymethyl)cyclobutyl]methyl}-1-(4-methoxyphenyl)urea
4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2-(propan-2-yl)-1,3-oxazole
1-[1-(3-methoxypropyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-5-{3-chloro-6-methylpyrazolo[1,5-a]pyrimidin-2-yl}-1H-1,2,4-triazole
2-({2-[4-(1H-imidazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)-4-methyl-5,6,7,8-tetrahydroquinazoline
1-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-(2-phenoxyethyl)piperazine
3-(3-{3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl)-1H-indole
5-methyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(1H-indazol-1-yl)-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
4-[1-(4-fluorophenyl)cyclopropanecarbonyl]-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
ethyl 3-[(2-fluorophenyl)methyl]-1-[4-(1H-1,2,4-triazol-1-yl)butanoyl]piperidine-3-carboxylate
N-cyclopropyl-3-[5-(oxolan-3-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
1-[3-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
methyl 5-{3-[4-(3-chlorophenyl)piperazin-1-yl]piperidin-1-yl}-5-oxopentanoate
2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}acetamide
5-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl]-1,2-dihydropyridin-2-one
4-benzyl-1-(3-chloro-2-fluorobenzoyl)-3-ethyl-1,4-diazepan-5-one
7-{1H-pyrrolo[2,3-b]pyridin-4-yl}-3,4-dihydro-2H-1-benzopyran-4-one
3-(1H-1,2,3-benzotriazol-4-yl)-1-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}urea
(3S,4S)-1-{2-[benzyl(methyl)amino]acetyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
3,5-difluoro-2-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]thiophene-3-carboxamide
2-benzyl-8-(3-fluoropropyl)-2,8-diazaspiro[5.5]undecan-3-one
2-{2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}-3-phenylcyclopent-2-en-1-one