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3-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[(4-fluorophenyl)methyl]-1,4-diazepan-5-one
N-methyl-3-(1H-pyrazol-4-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]propanamide
({4-[1-(3-fluorobenzoyl)piperidin-2-yl]phenyl}methyl)dimethylamine
4-[5-(1H-1,3-benzodiazol-2-yl)furan-2-yl]-N-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine
N-(1-benzylcyclopropyl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
6-[(diethylamino)methyl]-N-(1-methylpiperidin-4-yl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
1-tert-butyl-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidine-3-carboxamide
1-{[4-(5-methylfuran-2-yl)phenyl]methyl}-4-(1H-pyrrole-2-carbonyl)piperazine
2-(4-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}morpholin-3-yl)-N,N-dimethylacetamide
N-{2-[2-(methylcarbamoyl)ethyl]phenyl}-4-(morpholin-4-yl)piperidine-1-carboxamide
2-{4-[1-(2-methoxyethyl)piperidine-3-carbonyl]piperazin-1-yl}phenol
2-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]acetic acid
1-(cyclopropylmethyl)-N-ethyl-5-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]thiophene-3-carboxamide
1-(5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carbonyl)-4-ethylpiperazine
ethyl 1-{[5-(methoxymethyl)furan-2-yl]methyl}-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-methoxy-1-{1'-[2-(2-methylpiperidin-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-benzyl-3-(4-chlorobenzoyl)piperidine
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}oxane-2-carboxamide
ethyl 5-(1-{[(1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)pyridine-3-carboxylate
2,3-dimethyl-5-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]benzene-1-sulfonamide
3-[4-(adamantan-1-yl)piperazine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
1-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-4-(2-methoxybenzoyl)piperazine
(1R,6S)-3-[5-(4-methoxyphenyl)furan-2-carbonyl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane
2-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-5-chlorophenol
methyl 7-cyclohexyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxylate
2-(pyridin-3-ylmethyl)-9-(quinoxalin-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
7-methoxy-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-ethyl-1H-pyrazole-4-carboxamide
1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
N-(propan-2-yl)-1-[(1s,4s)-4-{[(3,4,5-trimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-methoxy-N-{1-[1-(naphthalen-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
3-methyl-N-{1-[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}butanamide
(1S,5R)-6-(cyclopropylmethyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-[(dimethylsulfamoyl)amino]-1-methyl-2-(2-methylpropyl)-N-(oxan-4-yl)-1H-1,3-benzodiazole-7-carboxamide
N-(oxan-4-yl)-3-(4H-1,2,4-triazol-4-yl)benzamide
6-(3-aminopyrrolidin-1-yl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[2-(3-oxopiperazin-1-yl)ethyl]benzamide
1-ethyl-3-methyl-N-{2-[(4-methylpyridin-2-yl)amino]ethyl}piperidine-3-carboxamide
N,N-dimethyl-2-(3-methylpentanamido)-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
methyl 2-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]piperidine-1-carboxylate
4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1,9-dimethyl-1,4,9-triazaspiro[5.6]dodecan-10-one
8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(2-phenylethyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-4-cyclopropyl-1-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)pyrrolidine-3-carboxylic acid
(3R,5S)-N-(adamantan-2-yl)-1-(propan-2-yl)-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
2-(3-methoxypropyl)-1-phenylmethanesulfonylpiperidine