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5-ethyl-N-[(1-ethyl-1H-imidazol-5-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
[(3R,4R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
N5-cyclopropyl-N6-(quinolin-6-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
{[(3R,4S)-1-(5-ethyl-2-methylpyrimidin-4-yl)-4-propylpyrrolidin-3-yl]sulfamoyl}dimethylamine
3-{[(1-hydroxy-2-methylpropan-2-yl)amino]methyl}-7-methyl-1-[(3-methylphenyl)methyl]-1,2-dihydroquinolin-2-one
ethyl 4-{[(6-chloropyridin-3-yl)carbamoyl]amino}piperidine-1-carboxylate
N-[(1-cyclohexylpiperidin-3-yl)methyl]-2-hydroxy-N-(pyridin-3-ylmethyl)acetamide
(2S,4R)-N,N-diethyl-4-[(1-methylpiperidin-4-yl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
2-{1-[1-(2,3-difluorobenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
4-{2-[(3-methoxyphenyl)carbamoyl]ethyl}-N-(2-phenylethyl)piperidine-1-carboxamide
(4aS,8aR)-6-(furan-3-carbonyl)-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
2-[5-(naphthalen-1-ylmethyl)-3-(propan-2-yl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-1-(2-ethylpiperidin-1-yl)propan-1-one
ethyl 5-(1-benzofuran-2-ylmethyl)-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(5-methyl-1,2-oxazol-3-yl)-5-[1-(1-methyl-1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-2-(pyrrolidin-1-yl)pyrimidine-5-carboxamide
2-(but-3-enoyl)-7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[(3S,4R)-1-[3-(benzyloxy)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
3-({3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
3-chloro-4-({1-[(4-ethylphenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
3,5-difluoro-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]pyridine-2-carboxamide
N-[2-(ethylsulfanyl)ethyl]-3-[(3-hydroxypiperidin-1-yl)sulfonyl]benzamide
2-(2-methoxyethyl)-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(thiophen-3-yl)phenoxy}acetamide
4-{1-[4-(pyrrolidin-1-yl)butanoyl]piperidin-3-yl}benzoic acid
(3R,4R)-4-(azepan-1-yl)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-3-ol
3-{1-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzamide
4-(5-methylpyridin-2-yl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperidin-4-ol
N-cyclopentyl-2-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]propanamide
5-{[3-(pyridin-2-ylmethoxy)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[(3R,4S)-1-[(2-cyanophenyl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
1-{[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl}piperidine-3-carbonitrile
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-4-(pyridin-4-yl)piperazine-1-carboxamide
11-(5-tert-butyl-1H-pyrazol-3-yl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
4-[3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carbonyl]-2,3-dihydro-1H-imidazol-2-one
4-(3,4-dimethoxyphenyl)-3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(2-{1-[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]piperidin-4-yl}ethyl)pyrrolidin-2-one
7-(furan-3-carbonyl)-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
5-methyl-6-(pyrrolidine-1-carbonyl)-N-[1-(thiophen-2-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
(1S,5R)-3-[2-(3,4-dimethylphenoxy)acetyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-methanesulfonylethan-1-one
3-{2-[4-(naphthalen-2-yl)piperazin-1-yl]-2-oxoethyl}-2,3-dihydro-1λ6-thiophene-1,1-dione
2-[3-(ethylsulfanyl)phenyl]-4-(pyrrolidine-1-carbonyl)pyridine
4-[4-(morpholine-4-carbonyl)piperidine-1-carbonyl]-5,6,7,8-tetrahydroquinazolin-2-amine
(4aR,7aS)-1-(2-methoxyacetyl)-4-[4-(thiophen-2-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(3R,4S)-1-[2-(2-methylphenyl)acetyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N,5-dimethyl-2-[1-(2-methylpropyl)-5-oxopyrrolidin-3-yl]-1H-imidazole-4-carboxamide