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3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-(3-ethylphenyl)piperidine-1-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]acetamide
2-{2-[4-(hydroxymethyl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-[1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-yl]pyrimidin-2-amine
2-(3-hydroxypropyl)-9-(2-phenylacetyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]azocane
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-(methylsulfanyl)-1,3-thiazole-4-carboxamide
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine
3-[2-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)-2-oxoethyl]-1,3-oxazolidin-2-one
4-{[5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-3-(3-fluorophenyl)piperazin-2-one
5-(4-phenylazepane-1-carbonyl)-1H-1,2,3-benzotriazole
8-{4-[(2-fluorophenyl)methoxy]benzoyl}-2,8-diazaspiro[4.5]decan-3-one
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3-cyclopropaneamido-4-methylbenzamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
2-methyl-5-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-3,4-dihydropyrimidin-4-one
[(3S,5R)-5-[(dimethylamino)methyl]-1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]piperidin-3-yl]methanol
1-(3-fluorophenyl)-3-{1-[1-(3-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
(1H-imidazol-4-ylmethyl)(methyl){2-[2-(prop-2-en-1-yl)phenoxy]ethyl}amine
4-[4-(1H-imidazol-2-yl)-1-phenyl-1H-pyrazol-3-yl]pyridine
1-(2-hydroxyethyl)-N-(1-phenylethyl)-5-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-(2-fluoroethyl)-3-[(3-phenoxyazetidin-1-yl)sulfonyl]benzamide
[(5-chloro-2-methoxyphenyl)methyl](ethyl)[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]amine
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(1-ethyl-1H-imidazol-2-yl)methyl]acetamide
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carboxamide
1-benzyl-5-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-yl}-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
ethyl[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
N-(4-methoxy-2-methylphenyl)-3-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}propanamide
N-(1-carbamoylcyclopentyl)-2-(4-fluorophenyl)imidazo[1,2-a]pyridine-6-carboxamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
5-{[4-(2-methanesulfonylethyl)piperazin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
3-chloro-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}thiophene-2-carboxamide
5-[benzyl(methyl)amino]-2-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
4-[4-(2-chlorophenyl)-2-methyl-5-oxopiperazin-1-yl]-4-oxobutanamide
3-[ethyl({[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl})amino]-1λ6-thiolane-1,1-dione
3-{[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]amino}pyrrolidin-2-one
2,5-dimethyl-3-{4-[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperazin-1-yl}pyrazine
5-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}-1,6-naphthyridine
2-(3-hydroxyadamantan-1-yl)-N-{2-[2-(trifluoromethyl)phenyl]ethyl}acetamide
N-({7-[3-(1,3-benzothiazol-2-yl)propanoyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methoxybenzamide
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-4-oxo-4-phenylbutanamide
[(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amine
5-[2-(3-methoxypropyl)piperidine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine
(1R,9S)-5-amino-3-(2,5-dimethoxyphenyl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
6-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidine-2,4-diamine
N-[(3-methoxyphenyl)methyl]-3-(N-methylmethanesulfonamido)-N-(prop-2-en-1-yl)propanamide
2-methyl-6-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
2-(cyclopropylmethyl)-9-(3,5-difluoropyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-methoxyphenyl)morpholine