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(2S)-2-amino-1-{4-[(4-fluorophenyl)methyl]piperidin-1-yl}-4-(methylsulfanyl)butan-1-one
2-methoxy-1-(1-methyl-4-{[2-(propan-2-yl)pyrimidin-5-yl]methyl}-1,4,9-triazaspiro[5.5]undecan-9-yl)ethan-1-one
(4-{[5-(1-ethyl-1H-1,2,4-triazol-5-yl)-4-phenyl-1H-imidazol-1-yl]methyl}phenyl)methanol
[3-propyl-1-(pyrimidin-2-ylmethyl)piperidin-3-yl]methanol
methyl 2-(quinolin-2-yl)benzoate
(1S,5R)-6-(5-chloro-2-fluorobenzoyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyrazin-2-amine
1-[(2,3-difluorophenyl)methyl]-4-[1-(4-methyl-1,3-oxazole-5-carbonyl)pyrrolidin-3-yl]piperidine
methyl 3-[(4-cyclohexanecarbonyl-7-oxo-1,4-diazepan-1-yl)methyl]benzoate
N-[2-(diethylamino)ethyl]-1-{2-[(3,4-dimethoxyphenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-ethylpiperidine-4-carboxamide
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(3,4-difluorophenyl)methyl]piperidine-3-carboxamide
2-[5-(2,3-dihydro-1,4-benzodioxin-2-yl)-1-(2-methylphenyl)-1H-1,2,4-triazol-3-yl]acetamide
N-[2-(azepan-1-yl)-2-phenylethyl]-3-(4-hydroxyphenyl)-1H-pyrazole-5-carboxamide
3-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
N-butyl-5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-methyl-1H-pyrazole-4-carboxamide
1-{4-fluoro-2-[3-methyl-1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}-1H-pyrazole
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2,3-dimethylquinoxaline-6-carboxamide
1-ethyl-N-(furan-3-ylmethyl)-N-methyl-5-[(3-methylbutyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
1-(cyclopropylmethyl)-5-(3-phenylpropyl)-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-cyclobutanecarbonyl-4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-({1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-2-yl}methyl)morpholine
1-(3,5-dimethylphenyl)-4-{5-[(methylsulfanyl)methyl]pyridin-2-yl}piperazin-2-one
2-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]phenoxymethyl}pyridine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[4-(1,3-thiazol-2-yl)piperazin-1-yl]ethan-1-one
1-[(5-methylfuran-2-yl)methyl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
4-(3-{[1-(2-phenylpropyl)piperidin-4-yl]oxy}benzoyl)morpholine
N-[(4-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethoxy}-3-methoxyphenyl)methyl]-N-[(3S)-2-oxoazepan-3-yl]cyclobutanecarboxamide
1-(4-methylphenyl)-4-[2-(piperidin-1-yl)acetyl]piperazin-2-one
2-(2-{[2-(2-fluorophenyl)ethyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
3-({2-[1-(4-methylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
5-[1-(4-chloro-2-methylphenyl)-1H-1,2,4-triazol-5-yl]-1-(2-methoxyethyl)piperidin-2-one
4-(4-chlorophenyl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]butanamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(4-methoxybenzoyl)piperidin-4-yl]propanamide
(2S)-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
2-methyl-N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)propanamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(methylsulfanyl)acetamide
8-(5-methylpyridine-3-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[(2-ethoxypyridin-3-yl)methyl]-4-methyl-3-(2-oxoimidazolidin-1-yl)benzamide
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-6-ethyl-2-(morpholin-4-yl)pyrimidin-4-amine
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-1-cycloheptyl-6-oxopiperidine-3-carboxamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4,4,4-trifluorobutan-1-one
4-(3-hydroxy-3-methylbutyl)-N-(2-methoxyethyl)-N-methylbenzamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-4-(1H-pyrazol-4-yl)butanamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1-benzofuran-2-carboxamide
1-[(5-ethylpyridin-2-yl)methyl]-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
(3-ethyl-1-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-3-yl)methanol
1-cyclopropyl-4-{[(5,6-dimethylpyrimidin-4-yl)amino]methyl}pyrrolidin-2-one