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5-{1-[(3-fluorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-1-methyl-1H-imidazole
3-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-3-[(dimethylamino)methyl]-3-(hydroxymethyl)piperidine-1-carboxamide
4-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1,3λ6,4-oxathiazinane-3,3-dione
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropylthiophene-2-carboxamide
3-[2-(1H-1,3-benzodiazol-1-yl)propanamido]-N-tert-butyl-2-methylbenzamide
4-(2-{3-[3-(2H-1,3-benzodioxol-5-yl)phenyl]-1H-pyrazol-1-yl}ethyl)morpholine
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-[3-(1H-imidazol-2-yl)propyl]-5-methylpiperidin-2-one
4-{1-[2-(3-chloro-2,6-difluorophenyl)-1H-imidazol-1-yl]propyl}pyridine
8-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1-[7-(1-hydroxy-3-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-methyl-1-oxobutan-2-yl}acetamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-5-methylthiophene-2-carboxamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-2-(1H-pyrazol-1-yl)butanamide
(2R,6R)-4-(2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}acetyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-(4-fluorophenyl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]butanamide
N-[(2-methoxyphenyl)methyl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-(pyridin-4-ylmethyl)propanamide
N5-(2H-1,3-benzodioxol-5-ylmethyl)-1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-(4-{[4-(1-hydroxyethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-2-(1H-pyrazol-1-yl)ethan-1-one
1-[(2-fluorophenyl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
(3S,4R)-4-(pyridin-3-yl)-1-(1,2,5-trimethyl-1H-pyrrole-3-carbonyl)pyrrolidine-3-carboxylic acid
2-(pyrrolidin-1-ylmethyl)-N-(3-sulfamoylphenyl)-1,4-oxazepane-4-carboxamide
3-(2-methoxypyrimidine-5-carbonyl)-3,9-diazaspiro[5.5]undecane
1-(4-fluorophenyl)-4-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]butane-1,4-dione
N-[2-(2-methoxyphenoxy)phenyl]-2,7-diazaspiro[4.5]decane-7-carboxamide
5-[1-methyl-5-(thiophen-2-yl)-1H-pyrazol-3-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
4-(4-fluorophenyl)-N-[(3-hydroxypyrrolidin-3-yl)methyl]oxane-4-carboxamide
3,7-dimethyl-11-[(6-methylpyridin-2-yl)methyl]-3,7,11-triazaspiro[5.6]dodecane
5-(dimethylamino)-2-[(3-phenylphenyl)methyl]-2,3-dihydropyridazin-3-one
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-2-cyclopropylacetamide
11-acetyl-4-[(5-methyl-1,2-oxazol-3-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N,N-dimethyl-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}propane-1-sulfonamide
6-methyl-3-{[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}-1,2-dihydroquinolin-2-one
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-(3-methoxypropyl)-1-(1,3-thiazol-4-ylmethyl)piperidine-3-carboxylic acid
4-{[2-(dimethylamino)ethyl]amino}-5-methyl-N-[3-(methylsulfanyl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-fluoroimidazo[1,2-a]pyridine-2-carboxamide
(1S,4S)-2-(2,5-dimethoxyphenyl)-5-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
4-(2-chlorophenoxy)-1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)piperidine
9-[6-(dimethylamino)pyrazin-2-yl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-[5-(2-amino-3-cyano-6-cyclopropylpyridin-4-yl)-2-methoxyphenoxy]acetic acid
3-[1-(1-cycloheptanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]propan-1-ol
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]benzamide
(4aS,7aR)-1-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[3-(pyridin-3-yl)propyl]piperidin-4-ol
(2S,4S)-1-benzyl-4-{[(4-chlorophenyl)methyl]amino}-N-ethylpyrrolidine-2-carboxamide
2-(3-{[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}phenoxy)acetamide
1-(4-methoxyphenyl)-5-methyl-4-[3-(pyridin-3-yl)propanoyl]piperazin-2-one
3-methyl-1-(2-methylpropyl)-4-(1,3-thiazol-4-ylmethyl)piperazin-2-one
(4aR,8aR)-7-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-carboxamide