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6-{4-[2-(1H-pyrazol-1-yl)butanoyl]piperazin-1-yl}pyridine-3-carbonitrile
(3R,4S)-4-cyclopropyl-1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-amine
N-[2-(3-fluorophenyl)ethyl]-6-oxo-1-(3-phenylpropyl)piperidine-3-carboxamide
4-(3-ethyl-1H-pyrazole-5-carbonyl)-1-(2-methoxyphenyl)piperazin-2-one
1-(1-methylpiperidin-4-yl)-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-[2-(cyclopropylmethyl)-4-[(oxolan-2-ylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
4-methyl-5-[1-(thiophen-3-ylmethyl)-1H-pyrazol-3-yl]-N-[(3,4,5-trifluorophenyl)methyl]-1,3-thiazol-2-amine
1-{2-[3-(benzyloxy)piperidin-1-yl]-2-oxoethyl}-3-methylimidazolidin-2-one
N-[3-(2,6-dimethylphenoxy)propyl]-N-methyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-[4-(4-fluorophenyl)-4-oxobutyl]-1,3-diazinane-2,4-dione
7-(2-methoxyethyl)-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-[3-(1H-imidazol-1-yl)phenyl]-4H-1,2,4-triazole
2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(trifluoromethyl)pyridine
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(5-methylfuran-2-yl)methyl]acetamide
(1R,5R)-6-benzyl-3-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-({1-[3-(2,3-dihydro-1H-isoindol-2-yl)propanoyl]pyrrolidin-3-yl}methyl)benzamide
1-[(4-chloro-3-fluorophenyl)methyl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
2-[2-chloro-6-methoxy-4-(thiomorpholin-4-ylmethyl)phenoxy]acetic acid
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-(1-methylpiperidin-3-yl)propanamide
N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-2-(4-methyl-1H-pyrazol-1-yl)acetamide
2-cyclopropyl-N,4-dimethyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidine-5-carboxamide
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-1-[3-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
8-[3-(1H-pyrazol-4-yl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{2-[(2,2-dimethyloxan-4-yl)formamido]ethyl}-N-[(4-methylphenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
methyl 2-{8-[(3-chloro-4-hydroxyphenyl)methyl]-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl}acetate
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(6-methyl-2-propylpyrimidin-4-yl)pyrrolidin-3-amine
N-(1,4-dioxan-2-ylmethyl)-1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-{3-oxo-2-azaspiro[4.5]decan-2-yl}acetamide
[2-(azepan-1-yl)ethyl](ethyl)(isoquinolin-5-ylmethyl)amine
2-(2-{[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-({5-[(2E)-2-methylbut-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-methylphenol
1-methyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-{2-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,2,3,4-tetrazole
(2S)-3-(3,3-diphenylpiperidin-1-yl)propane-1,2-diol
(1S,5R)-6-[(3,5-dimethyl-1H-indol-2-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
8-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-fluoro-N-methyl-2-oxo-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
9-(dimethyl-1,2-oxazole-4-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-1,1-dioxo-1λ6-thiolane-3-carboxamide
5-[(2R,3S,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridin-2-amine
N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-phenyl-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
(3S,4R)-4-(4-fluorophenyl)-1-[4-(2-oxopiperidin-1-yl)butanoyl]pyrrolidine-3-carboxylic acid
N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-5-methoxyfuran-2-carboxamide
N-[(2,4-difluorophenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-fluoro-4-[3-(2-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyridine
4-({5-[(1-ethylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
(3S,5R)-3-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-1-(2-methylpropyl)-5-(pyrrolidine-1-carbonyl)piperidine
2-benzyl-9-[2-(3-hydroxyphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one