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3-methyl-7-{2-methylthieno[3,2-d]pyrimidin-4-yl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
7-chloro-2-methyl-N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}quinoline-4-carboxamide
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(pyridin-3-yloxy)acetamide
(3-benzylpiperidin-3-yl)methanol
2-{[4-(4-methylphenyl)-5-(pyridin-3-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(2-{2-[1-(4-methoxy-2-methylbenzoyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
7-cyclopentyl-2-[3-(4-methyl-4H-1,2,4-triazol-3-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
5-methyl-N-(3-phenylpropyl)-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
[(3R,4R)-1-(7-methyl-1-benzofuran-2-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-methoxy-N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)benzamide
2-(3-methoxypropyl)-8-(1-methyl-1H-indole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1,9-dimethyl-4-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(oxolan-2-ylmethyl)-1-[1-(3-phenylpropanoyl)piperidin-4-yl]piperidine-4-carboxamide
3-tert-butyl-4-(7-methoxy-2H-1,3-benzodioxol-5-yl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[(2-aminopyrimidin-5-yl)methyl]-2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-methyl-1,3-oxazole-4-carboxamide
N-methyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
3-{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}-1,2-dihydropyridin-2-one
N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-3-[(3S,4R)-4-(morpholin-4-yl)-1-(pyridin-2-ylmethyl)piperidin-3-yl]propanamide
6-ethoxy-4-methyl-2-{3-[4-(pyrazin-2-yl)piperazine-1-carbonyl]piperidin-1-yl}quinazoline
dimethyl(3-{2-[1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
5-(4-fluorophenyl)-N-methyl-N-[3-(1H-pyrazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(pyridin-3-yl)ethan-1-one
4-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)piperidine-4-carboxylic acid
1-(5-chloronaphthalene-1-carbonyl)-4,4-difluoropiperidine
2-[4-(1H-indol-4-ylmethyl)piperazin-1-yl]-5-methyl-1,3-benzoxazole
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-[(4-phenylpiperazin-1-yl)methyl]piperidin-2-one
6-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-amine
4-[4-(2-methyl-1-benzothiophen-3-yl)-1H-imidazol-2-yl]-1-(pyridin-2-ylmethyl)pyrrolidin-2-one
2-{1-[(2-methylphenyl)methyl]-4-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperazin-2-yl}ethan-1-ol
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}cycloheptanecarboxamide
ethyl 1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
5-methyl-1-[(3-methylpyridin-2-yl)methyl]-5-phenylpiperidin-2-one
3-(3-fluoro-4-phenylbenzoyl)-N-propylpiperidine-1-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-[1-(pyridine-4-carbonyl)piperidin-4-yl]acetamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
(3R,4S)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-4-propylpyrrolidin-3-amine
2-{[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]methyl}benzonitrile
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[(3-methylpyridin-4-yl)methyl]amine
{[2-(methoxymethyl)pyrimidin-5-yl]methyl}(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
1-ethyl-1-(oxan-4-ylmethyl)-3-[2-(pyridin-3-yloxy)phenyl]urea
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
2-({6-[2-fluoro-3-(trifluoromethyl)phenyl]pyridazin-3-yl}(methyl)amino)ethan-1-ol
1-(3-chloro-4-methoxyphenyl)-N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-5-oxopyrrolidine-3-carboxamide
ethyl 4-[3-(2-amino-1,3-thiazol-4-yl)propanamido]piperidine-1-carboxylate
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(piperidin-1-yl)piperidine
(1R,5R)-6-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]-3-(thiophene-2-carbonyl)piperidine
N2-(2-methoxyethyl)-N4-[(5-methylpyrazin-2-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepane