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3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]propanamide
2-{4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-methyl-3-{3-[({2-[(4-methylphenyl)sulfanyl]ethyl}carbamoyl)amino]phenyl}propanamide
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-[methyl(propan-2-yl)amino]ethan-1-one
1-{1-[(3-fluorophenyl)methyl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
3-cyclopentyl-6-(oxolan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
9-(cyclopropylmethyl)-4-(3-fluoropropyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[5-({[(3-fluoro-4-methylphenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methyl-1,4-diazepan-1-yl)propan-2-ol
3-methyl-7-[1-(4-methylphenyl)cyclopropanecarbonyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N3-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-N5-butyl-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2,6,8-trimethylquinoline-4-carboxamide
2-[4-({4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]pyridine
2-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidin-1-yl]pyridine-3-carbonitrile
N-(3-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-3-oxopropyl)-N-methylmethanesulfonamide
5-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{4-[(5-chloro-3-methyl-1H-indol-2-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
2-(benzyloxy)-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]acetamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-(thiolan-3-yl)acetamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[2-(pyridin-3-yl)piperidin-1-yl]propan-1-one
methyl N-{[(3S,4S)-3-hydroxy-1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl]methyl}carbamate
(3S,4S)-1-(2-cyclopropyl-4-methylpyrimidine-5-carbonyl)-4-methylpiperidine-3,4-diol
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-(4-phenyl-1H-pyrazol-5-yl)piperidine
5-[1-(5-methyl-1,3-oxazole-4-carbonyl)pyrrolidin-2-yl]-N-(1,2,3-thiadiazol-5-yl)thiophene-2-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-(2-cyclopentanecarbonyl-1,2,3,4-tetrahydroisoquinolin-7-yl)-3-(4-methylphenyl)propanamide
4-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-2-methyl-1,4-oxazepane
2-methyl-5-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
6-[(4-ethyl-3,3-dimethylpiperazin-1-yl)methyl]pyridine-2-carboxylic acid
methyl 4-[5-({[(5-oxopyrrolidin-2-yl)methyl](propan-2-yl)amino}methyl)-1,2,4-oxadiazol-3-yl]benzoate
(3S,5R)-N3-(4-methylphenyl)-N5-[(1r,4r)-4-hydroxycyclohexyl]piperidine-3,5-dicarboxamide
3-(2-amino-1,3-thiazol-4-yl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}propanamide
N,N,4-trimethyl-3-{[methyl(prop-2-yn-1-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-benzyl-2-[1-(2-methoxyethyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}acetamide
5,8-dimethyl-2-{[4-(morpholine-4-carbonyl)piperazin-1-yl]methyl}quinolin-4-ol
N-(pyridin-2-ylmethyl)-1-[1-(pyridine-4-carbonyl)piperidin-4-yl]piperidine-3-carboxamide
1-cyclopentyl-5-{4-[(pyridin-2-yl)amino]piperidine-1-carbonyl}piperidin-2-one
3-[2-(2,4-difluorophenyl)ethyl]piperidine
7-(5-chloropyridin-2-yl)-4-[(2-fluorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2R,3R)-3-(dimethylamino)-1'-(1-methyl-1H-pyrazole-5-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N,N-dimethyl-5-[methyl(2-phenylethyl)amino]-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-cyclopentyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}urea
2-(2-{[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-{3-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]phenyl}ethan-1-one
(4aR,8aR)-2-methanesulfonyl-7-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
9-(1-methylcyclohexanecarbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-chloro-N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-indole-2-carboxamide
2-(4-fluoro-2-methoxyphenyl)-2-[(2-hydroxyethyl)(methyl)amino]acetic acid