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[1-(1H-indol-6-yl)-1H-1,3-benzodiazol-2-yl]methanol
2-[2-(dimethylamino)ethyl]-9-(3-fluorobenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
(1S,5R)-6-(5-methyl-1,2-oxazole-3-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
methyl 3-[4-({3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}methyl)-1H-pyrazol-1-yl]propanoate
1-[4-(quinazolin-4-yl)piperazin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
1-[(2,6-difluorophenyl)methyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
6-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
8-(1H-indazole-3-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(3-methoxypropyl)-8-(9H-purin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-benzyl-N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]pyrrolidin-3-amine
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
2-(dimethylamino)-1-[4-(ethoxymethyl)piperidin-1-yl]-2-(2-fluorophenyl)ethan-1-one
1-[2-(pyridin-4-yl)-4-{[2-(1H-pyrrol-1-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[4-(pyridin-2-yl)butyl]acetamide
1-[(2-methyl-1H-imidazol-4-yl)methyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
3-{2-oxo-2-[6-oxo-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]ethyl}imidazolidine-2,4-dione
2-(3-methyl-4-{spiro[indene-1,4'-piperidine]-1'-ylmethyl}-1H-pyrazol-1-yl)ethan-1-ol
4-[(4-fluorophenyl)methyl]-1-(furan-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]acetamide
2-{4-[(3-ethoxy-4-methoxyphenyl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidin-4-amine
2-(methylsulfanyl)-N-[(1S,3S)-3-{[4-(pyridin-3-yl)pyrimidin-2-yl]amino}cyclopentyl]acetamide
3-(2,4-difluorophenyl)-1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]propan-1-one
5-(5-oxopyrrolidine-2-carbonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[(2-butyl-4-methyl-3-oxopiperazin-1-yl)methyl]pyridine-3-carboxylic acid
3-ethyl-1-(3-methylbutyl)-8-[(6-methylpyridin-2-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(9aR)-2-methyl-8-(2-methylpropyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[(4-methoxyphenyl)methyl]-1-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-5-one
(4S)-3-{2-[4-(6-methylpyridin-2-yl)piperazin-1-yl]-2-oxoethyl}-4-phenyl-1,3-oxazolidin-2-one
5-{[4-(5-tert-butyl-1H-pyrazol-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-2-methoxypyrimidine
2-(4-methoxy-3-methylphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
N-(2-chlorophenyl)-3-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}propanamide
N3-(1,3-benzothiazol-2-ylmethyl)-N5-tert-butyl-1-cyclohexyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-4-({3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)phenol
1-methyl-N-(1-methylpiperidin-4-yl)-N-(2-phenylethyl)-1H-pyrrole-2-carboxamide
N-phenyl-3-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
N-[(5-methylpyrazin-2-yl)methyl]-5,6,7,8-tetrahydroquinoline-3-carboxamide
2-(3-chlorophenoxy)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)acetamide
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-3-(2-methoxyphenyl)propanamide
N-{[7-chloro-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)cyclohexanecarboxamide
4-[(3-methoxyphenyl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-benzyl-4-({4-[3-(methoxymethyl)piperidine-1-carbonyl]-1,3-oxazol-2-yl}methyl)piperazine
2-({6-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyrimidin-4-yl}amino)ethan-1-ol
2-{3-[3-(5-fluoro-2-methoxyphenyl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
1-(1-benzylpiperidin-4-yl)-N-(2-hydroxyethyl)piperidine-3-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[2-(1H-indol-3-yl)ethyl]propanamide
N,N-dimethyl-3-{[(2-methylphenyl)methyl]amino}-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)benzene-1-sulfonamide
4-[(2-{pyrazolo[1,5-a]pyrimidin-3-yl}phenyl)methyl]morpholine
2-methyl-5-{[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1,3,4-oxadiazole