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methyl 5-{[5-(oxan-2-yl)furan-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
ethyl 3-benzyl-1-(prop-2-ene-1-sulfonyl)piperidine-3-carboxylate
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-amine
N3-{3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]phenyl}piperidine-1,3-dicarboxamide
4-(2-fluorobenzoyl)-9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(3aR,6aR)-2-[(3,5-dimethoxyphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
7-{5-[(4-methylpiperidin-1-yl)methyl]furan-2-carbonyl}-2,7-diazaspiro[4.5]decane
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-4-(1-phenyl-1H-imidazol-4-yl)benzamide
N-[2-(ethanesulfonyl)ethyl]-3-(1H-1,2,4-triazol-1-yl)adamantane-1-carboxamide
3-{2-[1-(4-fluorophenyl)-3-phenyl-1H-1,2,4-triazol-5-yl]ethyl}oxolan-2-one
N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}-2-[4-(pyrazin-2-yl)-1H-pyrazol-1-yl]acetamide
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[2-(4-ethylmorpholin-2-yl)ethyl]-2-(furan-2-yl)-2-oxoacetamide
ethyl 1-ethyl-5-[3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-[2-({[(3S,4R)-4-hydroxyoxolan-3-yl](methyl)amino}methyl)-4-(thiophen-3-yl)phenoxy]acetic acid
5-cyclopropanecarbonyl-1'-[(2E)-3-phenylprop-2-en-1-yl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(1H-indol-4-ylmethyl)-3-(1H-pyrazol-1-yl)benzamide
1-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}pent-4-en-1-one
ethyl 4-{5-oxo-1,4,9-triazaspiro[5.5]undecan-9-yl}piperidine-1-carboxylate
3-(azepane-1-carbonyl)-N-ethyl-1-methyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-4-propyl-1,4-diazepan-5-one
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
(2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-{methyl[(methylcarbamoyl)methyl]carbamoyl}pyrrolidine-2-carboxylic acid
7-(3-methoxypropyl)-2-(1-methyl-1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
{[6-(4-fluorophenyl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(methyl)[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]amine
4-[(3-chloro-5-fluorophenyl)methyl]-2-ethyl-1-(propan-2-yl)piperazine
1-{1-[6-(2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carbonyl]piperidin-3-yl}-3-methylbutan-1-one
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,5R)-3-methanesulfonyl-6-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4S)-N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
methyl 4-(methylsulfanyl)-2-(3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamido)butanoate
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-3-{imidazo[1,2-a]pyridin-2-yl}propan-1-one
(2R)-2-{4-phenyl-5-[4-(pyrimidin-5-yl)phenyl]-1H-imidazol-1-yl}propanamide
N-[3-(4-fluorophenyl)phenyl]-1-(3-hydroxy-2,2-dimethylpropyl)piperidine-3-carboxamide
N-ethyl-5-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]pyrimidin-2-amine
1'-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]spiro[indene-1,4'-piperidine]
3-[2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-1,3-oxazolidin-2-one
4-(1-methylpiperidine-4-carbonyl)-1-(propan-2-yl)-6-{[4-(trifluoromethoxy)phenyl]methoxy}-1,4-diazepan-2-one
3-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-3,4-dihydropteridin-4-one
(2S)-3-(4-hydroxyphenyl)-2-[(1-methyl-1H-1,3-benzodiazol-5-yl)formamido]propanamide
N'1-[(3R,4S)-1-[(5-ethylpyridin-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
3-(2H-1,3-benzodioxol-5-yl)-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
methyl 2-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]acetate
4-(dimethyl-1,3-thiazole-4-amido)-N-phenylpiperidine-1-carboxamide
2-[4-(cyclopropylmethyl)piperazin-1-yl]-2-(2,6-dimethoxy-4-methylphenyl)acetic acid
8-{2-[ethyl(methyl)amino]acetyl}-3-(2-ethylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-methyl-2-oxo-8-(pyridine-2-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
8-chloro-2-[({2-[(3-methylpyridin-2-yl)amino]ethyl}amino)methyl]quinolin-4-ol
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amine
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-[(4-methylpiperazin-1-yl)methyl]piperidin-2-one