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4-{pyrazolo[1,5-a]pyridin-7-yl}pyridin-2-amine
N-[4-(3-methylphenyl)phenyl]-1-[2-(4H-1,2,4-triazol-4-yl)ethyl]piperidine-4-carboxamide
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)acetamide
5-[1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-4-yl]-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[(5-methyl-1H-imidazol-4-yl)methyl]benzamide
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]naphthalene-1-carboxamide
1-{2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-2,3-dihydro-1H-imidazol-2-one
3-(3-hydroxypyrrolidine-1-carbonyl)-1,4,6-trimethyl-1,2-dihydropyridin-2-one
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
4-{1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-4-yl}-5-(3-methoxyphenyl)-2-(pyridin-4-yl)pyrimidine
(3S,4R)-1-[2-(2-oxopyrrolidin-1-yl)ethyl]-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
4-ethyl-5-methyl-6-{9-oxa-2-azaspiro[5.5]undecan-2-yl}pyrimidin-2-amine
4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
2-{[1-(2-fluorophenyl)cyclopropyl]formamido}-N-(propan-2-yl)acetamide
4-(2-fluoro-3-methoxyphenyl)-6-methylpyrimidin-2-amine
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine-2-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)benzamide
4-[3-(2-chlorophenyl)pyrrolidine-1-carbonyl]-1-cyclohexyl-1H-1,2,3-triazole
3-cyclobutyl-5-[(2,5-dimethylthiophen-3-yl)sulfonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
6-{6-[3-(dimethylamino)propoxy]pyridin-3-yl}quinazolin-4-amine
5-[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]pyridin-3-amine
N-[(7S,8aS)-2-methyl-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-sulfamoylthiophene-2-carboxamide
2,3,6-trimethyl-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]quinoline-4-carboxamide
1-(carbamoylmethyl)-N-{[5-(dimethylcarbamoyl)furan-2-yl]methyl}piperidine-4-carboxamide
1-[(5-propylfuran-2-yl)methyl]-4-(1H-pyrazol-3-yl)piperidine
ethyl 4-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)piperidine-1-carboxylate
8-[3-(3-methoxy-4-methylphenyl)propanoyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3-(dimethyl-1,2-oxazol-4-yl)propanamide
1-[4-({3-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)phenyl]ethan-1-one
3-{5-[(4-methyl-1H-imidazol-5-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)-1-(thiophen-3-ylmethyl)piperidine
3-[1-({2-[(carboxymethyl)(methyl)amino]pyrimidin-5-yl}methyl)piperidin-3-yl]benzoic acid
{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}(methyl)(oxan-2-ylmethyl)amine
(2-{1-[(3-chloro-5-fluorophenyl)methyl]piperidin-2-yl}ethyl)dimethylamine
4-(1-{[1-(methoxymethyl)cyclopropyl]methyl}-4-phenyl-1H-imidazol-5-yl)phenol
2,7-dioxo-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,3-diazepane-4-carboxamide
(4aS,7aR)-1-[2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
2-amino-6-(6-methoxypyridin-3-yl)-4-[2-(propylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
N-[2-(3-methoxyphenyl)-1-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)ethyl]-N-methylfuran-2-carboxamide
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1-benzothiophene-2-carboxamide
2-[4-({4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}methyl)phenoxy]acetic acid
2-butyl-8-[(2,3-difluoro-6-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
4-(3-phenyl-1,2,4-oxadiazol-5-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}piperidine
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-4-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
(2S,4S,5R)-1-methyl-4-{[(3-methyl-1,2-oxazol-5-yl)methyl]carbamoyl}-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
1-({[(1R,2R)-2-(benzyloxy)cyclopentyl]carbamoyl}methyl)piperidine-4-carboxamide
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-(1-{1-[4-(1-benzofuran-2-yl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperidin-4-yl)piperidin-4-ol
N-[2,2-dimethyl-3-(morpholin-4-yl)propyl]-1H-indazol-5-amine