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9-hydroxy-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
ethyl 1-(4-hydroxy-2,3-dimethylphenyl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethan-1-one
N-[(4-fluorophenyl)methyl]-2,6-dioxo-N-(oxolan-2-ylmethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
(1S,5R)-6-(furan-2-carbonyl)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
3-(2-tert-butyl-6-methylphenyl)-1-[2-(1-methylpiperidin-3-yl)ethyl]urea
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-4-(2-phenylethyl)piperidine
(2S,4R)-4-amino-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-fluoro-2-[(2-methoxyphenyl)methyl]-1-[1-(oxolane-2-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2,2-dimethylthiomorpholin-3-one
N-pentyl-6-[(pyridin-3-yl)sulfamoyl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-2-(1H-pyrazol-1-yl)propan-1-one
3-(azepane-1-carbonyl)-2-[(3-fluorophenyl)methyl]-6-methyl-1-[3-(morpholin-4-yl)propyl]-1,4-dihydropyridin-4-one
2-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]quinoline-4-carboxylic acid
(2S,4R)-4-cyclopentaneamido-N,N-diethyl-1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidine-2-carboxamide
5-methyl-1-{2-oxo-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(3,4-dimethoxyphenyl)-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-amine
4-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-2-(4-methylpentyl)morpholine
6-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
5-(azocane-1-carbonyl)-1-cyclohexyl-N-cyclopropyl-4-oxo-1,4-dihydropyridine-3-carboxamide
1-{1-[(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)methyl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
2-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-4-methylphenol
2-[5-(4-fluoro-3-methylphenyl)-4-phenyl-1H-imidazol-1-yl]-N-methylbutanamide
1-{2-[(1-ethyl-1H-imidazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-7-yl}-3-phenylpropan-1-one
[(dimethyl-1,2-oxazol-4-yl)methyl](methyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
N-(furan-2-ylmethyl)-1-[4-(1-methyl-1H-1,2,4-triazol-5-yl)pyrimidin-2-yl]piperidine-4-carboxamide
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-(3,5-dichlorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-[3-(4-fluorophenyl)pyrrolidin-1-yl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
2-[methyl(pyridin-2-ylmethyl)amino]-1-(3-methyl-3-phenylpiperidin-1-yl)ethan-1-one
1-(2-methoxyacetyl)-N-[1-(pyridin-3-yl)pentyl]piperidine-4-carboxamide
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxane-4-carbonyl)piperidine
N,2-dimethyl-N-[1-(pyridin-2-yl)propan-2-yl]-2-(1H-pyrrol-1-yl)propanamide
(2S,3R)-2-amino-3-hydroxy-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
2-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-1-(thiolan-3-yl)-1H-imidazole
4-chloro-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,1-dimethyl-1H-indole-2-carboxamide
1-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-{4-[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]-1,4-diazepan-1-yl}ethan-1-one
2-[(4-benzylpiperazin-1-yl)methyl]-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-4-(4-ethoxy-3-methylphenyl)-4-oxobutanamide
4-{[(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)carbamoyl]amino}-N,3-dimethylbenzamide
6-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyridin-3-ol
4-{[4-(4-methoxyphenoxy)piperidin-1-yl]methyl}-1-methyl-1H-pyrrole-2-carbonitrile
4-phenyl-3-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}azetidin-3-yl)piperidine
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
ethyl 5-[({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)methyl]furan-2-carboxylate
({4-[(1-cyclohexanecarbonylpiperidin-3-yl)methoxy]phenyl}methyl)(methyl)[2-(pyridin-2-yl)ethyl]amine
3-[(1-methyl-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-amino-N-(2-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}ethyl)cyclobutane-1-carboxamide