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3-(5-ethylpyrimidin-2-yl)phenol
[(3R,4R)-1-[(3,5-dichloropyridin-4-yl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
(3R,5S)-N-[2-(1H-imidazol-4-yl)ethyl]-5-[(pyridin-3-yloxy)methyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
(3S,4R)-4-methyl-1-[3-(3-methylphenyl)-1H-pyrazole-4-carbonyl]piperidine-3,4-diol
2-methyl-6-[1-(1-phenylcyclopentanecarbonyl)piperidin-3-yl]pyrimidin-4-ol
N-[(2,3-dimethoxyphenyl)methyl]-1-(6-methoxypyrimidin-4-yl)piperidin-4-amine
2-ethoxy-5-(2-{[(5-methyl-1,2-oxazol-3-yl)methyl]amino}pyrimidin-4-yl)benzoic acid
methyl 2-(ethylsulfamoyl)-6-{[4-(trifluoromethyl)phenyl]methyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
methyl 3-(4-{[4-(naphthalen-2-yl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)propanoate
2-(2-methyl-1,3-thiazol-4-yl)-1-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]ethan-1-one
3-(3-fluorophenyl)-4-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)piperazin-2-one
1-[4-(4-fluorophenyl)-1,4-diazepan-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
2-(4-methylpentyl)-4-(pyridine-3-sulfonyl)morpholine
3-[2-(2-hydroxyethoxy)ethyl]-1-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
1-[2-(3-methoxyphenyl)piperidin-1-yl]-4-phenylbutane-1,2-dione
N-[2-(4-{[3-(1H-indol-3-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]benzamide
1-cyclopentyl-N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-5-oxopyrrolidine-3-carboxamide
N-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}pyrrolidine-1-sulfonamide
3-[5-(carbamoylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-{2-[2-(3-hydroxyphenyl)ethyl]piperidin-1-yl}-3-(pyridin-4-yl)propan-1-one
2-methyl-6-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]pyrimidin-4-amine
4,6-dimethyl-3-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}-1,2-dihydropyridin-2-one
(7S,8aS)-7-{2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}-2-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
6-(2-hydroxy-3-phenylpropyl)-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-{[(4-ethyl-1,3-thiazol-2-yl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-[1-(cyclohexylmethyl)-4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl]ethan-1-ol
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]propan-1-one
4-ethyl-3-{2-[2-(3-phenyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]ethyl}-4H-1,2,4-triazole
N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N,5-dimethyl-3-phenyl-1,2-oxazole-4-carboxamide
N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-3-{[(5-methylthiophen-2-yl)methyl]amino}benzamide
N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
3-(cyclopropylmethyl)-5-(2-phenylethyl)-5-(piperidin-4-yl)imidazolidine-2,4-dione
(butan-2-yl)(pyridin-3-ylmethyl)(thiophen-3-ylmethyl)amine
2-(6-methoxy-2,6-dimethylheptyl)-5-(1H-1,2,3,4-tetrazol-1-yl)-1H-1,3-benzodiazole
1-(4-cyanopyridin-2-yl)-N-[4-(pyridin-3-yloxy)phenyl]piperidine-4-carboxamide
1-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-3-[(3-methyloxetan-3-yl)methyl]urea
3-[2-(azepan-1-yl)-2-oxoethyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-one
4-{4-[(4-methylpiperazin-1-yl)methyl]piperidine-1-carbonyl}-6-(propan-2-yl)pyrimidin-2-amine
N-(1-carbamoylcycloheptyl)-2,5-dimethyl-1,3-thiazole-4-carboxamide
N4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N4-methylpyrimidine-4,6-diamine
1-methyl-4-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,4-diazepane
1-benzyl-N-methyl-5-(pyrrolidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-(1'-{4-[ethyl(methyl)amino]pyrimidin-2-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)propan-1-one
2-{4-[(5-cyclohexylthiophen-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
2-(2-{[methyl(oxan-4-ylmethyl)amino]methyl}phenoxy)propanoic acid
3-[2-(3-methoxyphenyl)pyrrolidine-1-carbonyl]-6-methyl-4H-pyrido[1,2-a]pyrimidin-4-one
4-{2-[3-(2-methylpropyl)morpholin-4-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
3-(azepane-1-carbonyl)-1-ethyl-5-(piperidin-1-yl)-4,5,6,7-tetrahydro-1H-indazole
(2R,6R)-4-[4-(2-oxopyrrolidin-1-yl)butanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3,3,3-trifluoropropanamide