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N4-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-6-methylpyrimidine-2,4-diamine
1-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-3-(propan-2-yl)urea
7-methoxy-3-{[3-(methoxymethyl)piperidin-1-yl]sulfonyl}-2,3,4,5-tetrahydro-1H-3-benzazepine
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-[(2-methoxypyrimidin-5-yl)methyl]piperidin-4-ol
3-[4-(3-methylphenyl)piperazin-1-yl]-N-[3-(pyridin-2-yl)propyl]propanamide
1-{3-[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]-3-oxopropyl}pyrrolidin-2-one
[(3S,5R)-1-(3-chlorothiophene-2-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}acetamide
4-(cyclopropylmethyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-3-(propan-2-yl)-1,4-diazepan-5-one
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
(3aS,6aS)-2-methyl-5-({5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoic acid
1-{1-[2-(1H-imidazol-1-yl)acetyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-3-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[2-(azepan-1-yl)-2-phenylethyl]-2-(2-oxopiperidin-1-yl)acetamide
(4aS,8aR)-6-(4-chloro-2-hydroxybenzoyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
3-[(cyclopentylamino)methyl]-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
4-chloro-1,3-dimethyl-N-[2-(phenylsulfanyl)ethyl]-1H-pyrazole-5-carboxamide
4-{1-[2-(3-oxopiperazin-1-yl)acetyl]piperidin-3-yl}benzoic acid
1-methyl-9-(prop-2-en-1-yl)-4-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-cyclopropyl-2-(3-acetamidophenyl)pyridine-4-carboxamide
6-methyl-2-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]-4-(thiophen-2-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
1-(propan-2-yl)-4-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
2-[(adamantan-1-ylmethyl)({[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})amino]ethan-1-ol
(1R,5R)-6-benzyl-3-(thiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-1-(1H-indole-2-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
7-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3-(2-acetamidoacetamido)-4-(2-methylpiperidin-1-yl)benzamide
(4aR,7aS)-1-acetyl-4-(1H-indole-6-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(3-{4-[(1H-imidazol-2-ylmethyl)amino]piperidin-1-yl}phenyl)-3-methylimidazolidin-2-one
1-methanesulfonyl-4-(3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}phenoxy)piperidine
N-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]azocane-1-carboxamide
1-(4-fluorophenyl)-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,4-diazepane
1-(2-ethoxyethyl)-N-[(4-hydroxyphenyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-4-yl)-1,2,3,4-tetrahydroisoquinoline
methyl 3-[(3S,4R)-1-cycloheptyl-4-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-3-yl]propanoate
2-({[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amino}methyl)benzoic acid
2-[3-(ethylsulfanyl)phenyl]-4-(piperidine-1-carbonyl)pyridine
5-(oxolane-3-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-[(2-ethyl-6-methylpyridin-3-yl)oxy]-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-methyl-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperazine
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[(3-fluorophenyl)methyl]piperidin-3-ol
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(1H-pyrazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3S,4R)-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazine
3-(2,6-dimethylphenoxy)-1-{imidazo[1,2-a]pyridine-6-carbonyl}azetidine
6-(piperidin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
1-[(4-fluorophenyl)methyl]-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide