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1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3S,4R)-4-(3-fluorophenyl)-1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]pyrrolidine-3-carboxylic acid
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[4-(pyrimidin-2-yloxy)phenyl]methyl}piperidin-3-ol
4-[(2-hydroxyethyl)sulfamoyl]-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]benzamide
N3-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-N1,N1-dimethylpiperidine-1,3-dicarboxamide
4-{5-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]furan-2-yl}-2-methylbut-3-yn-2-ol
(1S,5R)-6-(pyridin-2-ylmethyl)-3-[(2,3,4-trifluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
4-{2-[4-(2-methoxyethyl)phenoxymethyl]phenyl}-6-methyl-2,3-dihydropyridazin-3-one
6-[4-(2-methoxyethoxy)phenyl]-2-methyl-1H-imidazo[4,5-b]pyridine
2-(5,5-dimethyl-2,4-dioxo-1,3-oxazolidin-3-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
2-(4-chloro-2-methoxybenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-methyl-2-[4-(morpholin-4-yl)-2-(thiomorpholin-4-yl)pyrimidin-5-yl]propanoic acid
(3R,4R)-3-methyl-1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-(oxan-4-yl)piperidin-4-ol
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-methyl-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)urea
methyl (2S,4R)-4-(2,2-diphenylacetamido)-1-[(4-hydroxy-3-methoxyphenyl)methyl]pyrrolidine-2-carboxylate
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-amine
4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(4-methyl-1H-imidazole-2-carbonyl)piperidine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-N'-(2-fluoro-5-methylphenyl)butanediamide
methyl 2-cyclopropyl-1H-1,3-benzodiazole-6-carboxylate
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
5-chloro-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-fluoro-N-methylpyridin-2-amine
4-[6-(2-butoxy-4-fluorophenyl)pyridine-3-carbonyl]morpholine
1-(5-methoxy-2-{[(quinolin-3-ylmethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
N-cyclohexyl-5-(1-{[(2-ethylpyrimidin-5-yl)methyl]amino}ethyl)-N,4-dimethylpyrimidin-2-amine
N-[(4-fluorophenyl)methyl]-3-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}propanamide
(2R)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}-5-oxopyrrolidine-2-carboxamide
N-cyclobutyl-2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
8-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-N-phenylpiperidin-3-amine
3-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]-6-(propan-2-yl)pyridazine
1-methanesulfonyl-4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-1,4-diazepane
2-ethyl-9-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-phenyl-2,9-diazaspiro[5.5]undecane
4-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}pyridin-1-ium-1-olate
2-(4-hydroxypiperidin-1-yl)-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-6-[4-(methylsulfanyl)phenyl]pyridine-3-carboxamide
(2S,4S)-N-ethyl-1-(oxan-4-yl)-4-(3-phenylpropanamido)pyrrolidine-2-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-benzyl-1-(4-methoxyphenyl)-4-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl({[1-(2-methylpropyl)-2-phenylmethanesulfonyl-1H-imidazol-5-yl]methyl})[2-(1H-pyrazol-4-yl)ethyl]amine
5-[4-(2-ethoxyphenyl)piperazine-1-carbonyl]-1-[(3-fluorophenyl)methyl]piperidin-2-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
9-(oxolan-3-ylmethoxy)-4-(pyridine-2-carbonyl)-7-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[(dimethylsulfamoyl)amino]-1-(naphthalen-1-ylmethyl)pyrrolidin-2-one
(4aR,7aS)-1-(2-methoxyethyl)-4-[(2-methyl-1,3-thiazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(furan-2-carbonyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
N-(2-{4-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]morpholin-2-yl}ethyl)acetamide
1-cyclopropanecarbonyl-4-{4-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]phenoxy}piperidine
N-{3-methyl-1-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]butyl}thiophene-2-carboxamide
3-[(3R,4S)-1-[3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
N-{2-[(4-chlorophenyl)methoxy]ethyl}-2-(hydroxymethyl)-1H-1,3-benzodiazole-5-carboxamide
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one