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2-amino-4-cyclopropyl-6-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]pyridine-3-carbonitrile
[1-(2-aminopyridin-4-yl)-3-(cyclopropylmethyl)piperidin-3-yl]methanol
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-{2-[(3-methoxyphenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidine
8-chloro-3-(1-hydroxypropan-2-yl)-3,4-dihydroquinazolin-4-one
N-[2-(morpholin-4-ylmethyl)phenyl]-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
8-(4-aminocyclohexyl)-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
3-(2,3-dimethoxyphenyl)-N-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
N-(1-cycloheptylpiperidin-3-yl)-1-ethyl-3-methyl-1H-pyrazole-4-sulfonamide
N-[(5-chloro-1H-1,3-benzodiazol-2-yl)methyl]-8-fluoro-N-methylquinoline-2-carboxamide
2-(3-fluorophenoxymethyl)-8-(5-methylpyridine-3-carbonyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-(pyrrolidin-3-yl)piperazine
(1R,3S,5S)-8-{5-ethyl-6-methylthieno[2,3-d]pyrimidin-4-yl}-8-azabicyclo[3.2.1]octan-3-ol
N-[(5-amino-1,3,4-thiadiazol-2-yl)(phenyl)methyl]-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
1-(azepane-1-sulfonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-(6-methoxynaphthalene-2-carbonyl)-1-(1-methylpiperidin-4-yl)piperidine
(1R,5R)-6-(3-{[(4-fluorophenyl)methyl]sulfanyl}propanoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-methyl-8-[(1-methyl-1H-indol-6-yl)methyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
5-[2-(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)-2-oxoethyl]-2-methyl-3,4-dihydropyrimidin-4-one
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
6-tert-butyl-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3S,4S)-1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}piperidine-3,4-diol
N-(4-fluoro-3-{[(2-methoxyethyl)(1-methylpiperidin-4-yl)carbamoyl]amino}phenyl)propanamide
(4aS,8aS)-2-(6-chloro-8-methylquinolin-4-yl)-decahydro-2,7-naphthyridin-4a-ol
2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
4-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}morpholine
2-chloro-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
5,7-dimethyl-N-[1-(1H-pyrazol-1-yl)propan-2-yl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
2-[methyl({4-methyl-5-[1-(pyridin-4-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
3-(1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}piperidin-4-yl)-N-(2-methoxyethyl)propanamide
4-phenyl-2-[4-(5-propyl-1,2-oxazole-3-carbonyl)piperazin-1-yl]pyrimidine
1-[4-(difluoromethoxy)benzoyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
(1S,5R)-3-(pyridine-3-carbonyl)-6-(1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,5R)-1-[5-(ethylsulfanyl)thiophene-2-carbonyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
3-[({1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
2-({3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}methyl)pyridine-3-carboxylic acid
1-[2-(cyclohexylcarbamoyl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
6-(4-{7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carbonyl}piperazin-1-yl)pyridine-3-carbonitrile
5-(4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)-1H-imidazol-2-amine
({2-[(2-chlorophenyl)methoxy]-6-methylquinolin-3-yl}methyl)[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]amine
4-hydroxy-2-methyl-N-[1-(oxan-4-yl)piperidin-4-yl]pyrimidine-5-carboxamide
5-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyrazin-2-ol
5-methyl-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1-(pyridin-2-yl)-1H-pyrazole-4-carboxamide
3-[(3R,4S)-3-[3-(5-methyl-1H-1,2,4-triazol-3-yl)propanamido]-4-(propan-2-yl)pyrrolidin-1-yl]propanoic acid
methyl 4-({2-[(3-methoxyphenyl)methyl]morpholin-4-yl}methyl)benzoate
3-methyl-3-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[3-(4-methylpiperazine-1-carbonyl)phenyl]urea
3-(1-{1-[(4-chlorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
2-(cyclobutylmethyl)-5-(4-methylpiperazin-1-yl)-2,3-dihydropyridazin-3-one
(3R,4R)-1-(3-chloropyridin-2-yl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
(3S,7S)-5-(5-cyclopropyl-3-methyl-1H-pyrazole-4-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid