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8-{[2-(methylsulfanyl)-5-oxo-5H-[1,3,4]thiadiazolo[3,2-a]pyrimidin-7-yl]methyl}-2,8-diazaspiro[4.5]decan-3-one
4-[(1-ethylpyrrolidin-3-yl)methyl]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
9-methoxy-7-(5-methylthiophen-2-yl)-4-(quinolin-8-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
8-chloro-N-(1-ethoxy-2-methylpropan-2-yl)quinoline-2-carboxamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)pyrazolo[1,5-a]pyridine-7-carboxamide
methyl 3-cyclohexyl-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate
(1H-imidazol-2-ylmethyl)(methyl)[(2-methyl-2,3-dihydro-1-benzofuran-5-yl)methyl]amine
2-[3-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)phenoxy]acetamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-(3-hydroxyquinoxalin-2-yl)propanamide
2-(2,4-dimethoxyphenyl)-2-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}acetic acid
1-{4-[(4-fluoropiperidin-1-yl)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)imidazo[1,2-a]pyridine-6-carboxamide
4-ethyl-1-[(4-fluorophenyl)methyl]-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-4-amino-N-ethyl-1-[3-(4-oxo-3,4-dihydroquinazolin-3-yl)propanoyl]pyrrolidine-2-carboxamide
N,N-diethyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-(1-{2-[methyl(pyridin-2-ylmethyl)amino]acetyl}piperidin-3-yl)benzoic acid
N-[2-(4-fluorophenyl)ethyl]-N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}cyclopropanecarboxamide
(3S,4S)-1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(naphthalen-2-yl)piperidin-3-ol
(2R,3R,6R)-N,N-dimethyl-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-sulfonamide
6-ethyl-4-[2-(thiophen-2-yl)azetidine-1-carbonyl]-1,2-dihydropyridin-2-one
4-[(2-methyl-1H-imidazol-4-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
8-(2,3-difluoro-4-methylbenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(4,6-dimethylquinolin-2-yl)amino]-N-ethylpiperidine-1-carboxamide
3-(1,3-diethyl-6-methyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
5-[1-(3,4-dimethoxyphenyl)-1H-imidazol-2-yl]-N,N-dimethylpyrimidin-2-amine
7-ethoxy-4-(isoquinolin-5-yl)-1,2,3,4-tetrahydroquinolin-2-one
N,1-dimethyl-N-[(1-methylpyrrolidin-3-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2-{1-[3-(benzylsulfanyl)propanoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
4-{4-[(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)methyl]phenyl}-2-methylbut-3-yn-2-ol
3-{7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-N,N-dimethylaniline
4-(1-ethyl-1H-pyrazole-3-carbonyl)-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(2,5-dichlorophenyl)-1-[1-(pyrazin-2-yl)piperidin-3-yl]urea
N-(3-methoxypropyl)-1-methyl-N-[(1-methyl-1H-indol-2-yl)methyl]piperidin-4-amine
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(2,2-dimethylpropyl)propanamide
ethyl[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}amine
2-(5-amino-4H-1,2,4-triazol-3-yl)-N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)acetamide
6-ethyl-N-[2-(3-methoxyphenoxy)ethyl]-N-methylpyrimidin-4-amine
5-{4-[3-(1-methoxyethyl)phenyl]-1H-pyrazol-1-yl}-1H-1,2,3,4-tetrazole
(3aS,6aS)-2-benzyl-5-(1H-imidazole-5-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(6-ethylpyrimidin-4-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
methyl 2-{1-methyl-2-oxo-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}acetate
2-{2-[4-(2,2-dimethyloxan-4-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,3-benzodiazole
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}pyrimidin-2-amine
1-[2-(1-cycloheptylpiperidin-3-yl)ethyl]-3-(propan-2-yl)urea
5-(3-oxo-4-phenylpiperazine-1-carbonyl)pyridine-2-carbonitrile
1-{2-[3-(3-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}piperidin-2-one
1-benzyl-3-(2-methylphenyl)-3-{2-oxo-2-[4-(pyrazin-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
1-(difluoromethyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrazole-3-carboxamide
(1-{2-[5-(3-methylthiophen-2-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-3-yl)methanol