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N-[2-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propyl]-2-(morpholin-3-yl)acetamide
N-(2-phenylethyl)-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-(3-fluoro-2-methylphenyl)acetamide
3-[(3R,4S)-1-[(3,5-dichloropyridin-4-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
3-hydroxy-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyridine-2-carboxamide
2-{4-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[2-(cyclohexylsulfanyl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
7-[(2R)-2-cyclohexyl-2-hydroxyacetyl]-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(2-oxoimidazolidin-1-yl)-N-[2-(pyridin-2-ylsulfanyl)ethyl]benzamide
{1-[1-(2,3-dimethyl-1H-indole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}(methyl)(pyridin-4-ylmethyl)amine
1-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-{[4-(1H-imidazol-2-yl)piperidin-1-yl]methyl}-8-methoxyquinoline
N-benzyl-1,3-dimethyl-N-(oxolan-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-amino-6-[4-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperazin-1-yl]pyrimidin-4-ol
2-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-1-(4-methylpiperazin-1-yl)ethan-1-one
(1R,5S,6R)-3-[(2-chloro-6-fluorophenyl)methyl]-N-(pyridin-2-ylmethyl)-3-azabicyclo[3.1.0]hexane-6-carboxamide
(1S,5R)-6-(furan-3-carbonyl)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
7-({methyl[3-(1H-pyrazol-1-yl)propyl]amino}methyl)-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
5-ethyl-2-methyl-4-{4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyrimidine
1-(cyclopropylmethyl)-6-(1-ethylpiperidin-4-yl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-({1-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]piperidin-3-yl}methyl)-1,3-thiazole-5-carboxamide
N-(3-{[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]sulfonyl}phenyl)acetamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
1-[3-(3-fluorophenyl)phenyl]-3-[2-(2-methylpropanesulfonyl)ethyl]urea
(4aS,7aR)-1-[(3-hydroxyphenyl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(1,3-benzothiazol-2-yl)-N-[2,2-dimethyl-3-(morpholin-4-yl)propyl]piperidin-3-amine
N-(1-hydroxybutan-2-yl)-4-methyl-N-[(2-methylphenyl)methyl]piperidine-4-carboxamide
3-[(tert-butylcarbamoyl)methyl]-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(hydroxymethyl)-N-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]piperidine-1-carboxamide
1-(4-methyl-2-{[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]amino}pyrimidin-5-yl)ethan-1-one
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
1-(2-fluorophenyl)-4-{1-[(2-methoxyphenyl)methyl]piperidin-3-yl}piperazine
N-[2-(dimethylsulfamoyl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
N-cyclobutyl-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-ethyl-4-phenyl-9-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
6-methyl-1-[3-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)propyl]-1,2-dihydropyridin-2-one
4-(4-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
N-[1-(1-{[3-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2-phenylacetamide
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(oxan-3-ylmethyl)pyridin-2-amine
4-ethyl-3-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methyl)-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(pyridin-4-ylmethyl)-4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1,4-diazepane
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(1-ethyl-1H-imidazol-2-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,4-dihydroquinolin-4-one
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
3,4,7-trimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-indole-2-carboxamide
1-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethan-1-one
1-methyl-3-propyl-N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-1H-pyrazole-5-carboxamide
9-(2,3-dimethoxyphenyl)-1-ethyl-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione