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N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-(thiomorpholine-4-sulfonyl)benzamide
3-(azepane-1-carbonyl)-1-ethyl-5-[4-(piperidin-1-yl)piperidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole
4-(4-methyl-1H-pyrazol-3-yl)-1-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperidine
6-ethoxy-3-({methyl[(1-methylpyrrolidin-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-{4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperazin-1-yl}pyrazine
1-[2-(adamantan-1-yl)-4-hydroxypyrimidine-5-carbonyl]piperidine-3-carbonitrile
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(3-chloro-4-fluorobenzoyl)pyrrolidin-3-yl]methanol
dimethyl({2-[4-(thiophene-3-carbonyl)morpholin-2-yl]ethyl})amine
4-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-6-methylpyrimidin-2-amine
7-(2-methoxyphenyl)-2-(3-methylpyridin-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
6-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carbonitrile
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)oxan-4-amine
1-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-N-(pyridin-3-ylmethyl)piperidin-4-amine
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
4-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1,5-dimethyl-1H-pyrazole
3-[1-(2-hydroxybutyl)-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]-1-methyl-1,4-dihydroquinolin-4-one
3-[(5-methoxy-4-oxo-4H-pyran-2-yl)methyl]-5-(piperidin-4-yl)-5-propylimidazolidine-2,4-dione
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(4-fluoro-3-methoxyphenyl)pyridine-3-carbonitrile
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-cyclopropyl-N-(1,3-thiazol-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
5-methyl-N-[1-(thian-4-yl)piperidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
methyl[(4-methyl-1H-imidazol-2-yl)methyl][(2,6,8-trimethylquinolin-4-yl)methyl]amine
{3-[(dimethylamino)methyl]-1-(furan-3-ylmethyl)piperidin-3-yl}methanol
2-{4-[(dimethylamino)methyl]phenyl}-N-(isoquinolin-5-yl)piperidine-1-carboxamide
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]propanamide
N-(2-methoxyethyl)-2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(1-ethyl-1H-1,2,4-triazol-3-yl)urea
4-(2,4-dioxoimidazolidin-1-yl)-N-(3-hydroxy-3-phenylpropyl)-N-methylbenzamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetamide
3-[(3-cyclohexyl-1,2-oxazol-5-yl)methyl]-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-oxo-1-(2-phenylethyl)piperidine-3-carboxamide
N-methyl-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
3-cyclopropyl-5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-1,2,4-triazole
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-1H-1,2,3-triazole-5-carboxamide
8-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
3-(1H-imidazol-1-yl)-1-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}propan-1-one
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
1-(4-fluorophenyl)-4-[1-(1H-pyrrole-2-carbonyl)piperidin-3-yl]piperazine
2-[({5-[1-(5-fluoropyridine-3-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
7-methyl-2-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,7-diazaspiro[4.5]decan-6-one
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-[methyl(pyridin-3-ylmethyl)amino]ethan-1-one
2-[3-(dimethylamino)propyl]-9-[(5-fluoro-2-methoxyphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-(1-cyclopentylpiperidine-3-carbonyl)-4-(pyrimidin-2-yl)-1,4-diazepane
1-(3-methylbutan-2-yl)-5-(pentan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
4-[5-(piperidine-1-carbonyl)pyridin-2-yl]-2-(trifluoromethyl)morpholine
3-(1H-imidazol-1-ylmethyl)-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
4-[3-cyclopropyl-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-3-fluoropyridine
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4-(5-methylpyridin-2-yl)piperidin-4-ol