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3-[(4-fluorophenyl)methyl]-N-(1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-(morpholin-2-yl)acetamide
4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]-N-[2-(pyrrolidin-1-yl)ethyl]benzamide
(3R,4R)-3-[(dimethylamino)methyl]-N-[2-(2-fluorophenyl)ethyl]-4-(hydroxymethyl)pyrrolidine-1-carboxamide
N-ethyl-7-fluoro-3-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-indole-2-carboxamide
methyl (2R,4S)-1-[5-(2-chlorophenyl)furan-2-carbonyl]-4-hydroxypiperidine-2-carboxylate
(3R,4R)-1-(4-aminopyrimidin-2-yl)-4-cyclobutyl-3-methylpiperidin-4-ol
N-{[2-(dimethylamino)pyridin-3-yl]methyl}-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
(3S,9aR)-3-benzyl-8-(quinolin-6-ylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3S,4R)-1-(2-ethoxybenzoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]-N-[1-(pyridin-4-yl)propan-2-yl]pyridin-2-amine
[(4-{1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-2-yl}phenyl)methyl]dimethylamine
3-[5-(pyridin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(1H-imidazol-1-yl)propan-1-one
1-(5-chloro-2-methoxyphenyl)-3-methyl-5-[(5-methyl-1H-pyrazol-1-yl)methyl]-1H-1,2,4-triazole
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-3-(pyrrolidine-1-carbonyl)benzene-1-sulfonamide
N-[1-(2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-4-yl]methanesulfonamide
3-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[(3-fluorophenyl)methyl]urea
N-[4-({[(4-fluorophenyl)methyl](oxolan-2-ylmethyl)amino}methyl)phenyl]acetamide
1-{2-[4-(2-fluorophenyl)piperazin-1-yl]-6-(2-methoxyphenyl)pyridine-3-carbonyl}piperidin-3-ol
2-{[1-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
1-{5-[(4-methylphenyl)methanesulfonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidine
1-(1-methylpiperidin-4-yl)-4-(1,3-thiazol-2-ylmethyl)piperazine
1-(1-{1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
N-(3-phenylprop-2-yn-1-yl)-N-(prop-2-en-1-yl)-1H-pyrrole-2-carboxamide
7-{4-[(dipropylamino)methyl]benzoyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}amine
2-(3-chlorophenoxy)-N-({8-[(2-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)propanamide
1-(2-fluorophenyl)-4-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
4-{[5-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)-1,2,4-oxadiazol-3-yl]methyl}morpholine
3-(3,5-dimethyl-1H-pyrazol-4-yl)-6-(4-methylpiperazin-1-yl)pyridazine
[(2S,6S)-4-(2-methyl-1,3-benzoxazole-6-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
5-{[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-N-propylpyrimidin-2-amine
({5-[1-(4-cyclobutyl-6-methylpyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-{[(2R,5S)-5-[(3-fluoro-4-methoxyphenyl)methyl]oxolan-2-yl]methyl}piperidine-4-carboxylic acid
[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl](methyl){[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
3-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
7-(6-methyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-{4-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
6-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-2-carbonitrile
2-tert-butyl-N-(5,6-dimethylpyrimidin-4-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-amine
2-[({1-azabicyclo[2.2.2]octan-3-yl}amino)methyl]-4-(6-methoxypyridin-2-yl)phenol
5-(4-cyclopentylpiperazin-1-yl)-N-[(4-fluorophenyl)methyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
6-[4-(azepan-1-yl)butyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-(2-methyl-6-{1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-4-yl}pyrimidin-4-yl)morpholine
N-[(2-methoxyphenyl)methyl]-N-(pyridin-3-ylmethyl)thiophene-3-carboxamide
N-[2-(5-hydroxypyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]pyridine-2-carboxamide
2-cyclopentyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one