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methyl (2R,4S)-4-hydroxy-1-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]piperidine-2-carboxylate
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-N-methylacetamide
2-{cyclopropyl[(3-methylthiophen-2-yl)methyl]amino}-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
1-{4-[1-(furan-2-ylmethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}-1H-1,2,4-triazole
1-methyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(2S,4R)-1-(2-chloro-4-fluorobenzoyl)-N-ethyl-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
1-benzyl-N-(1H-indol-3-yl)-1H-pyrazole-4-carboxamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(2-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
4-{[1-(1-methoxypropan-2-yl)piperidin-4-yl]oxy}-N-(pyridin-4-ylmethyl)benzamide
5-(5-hydroxypyrazine-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
1-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-3-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
4'-[(4-ethenylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-[(5-methylpyrazin-2-yl)methyl]-9-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-3-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}-4,5,6,7-tetrahydro-1H-indazole
N-[(1S,2R)-2-aminocyclobutyl]-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-3-sulfamoylthiophene-2-carboxamide
2-[2-(2-hydroxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carbonyl]benzonitrile
(1S,5R)-6-[(2-cyclohexylpyrimidin-5-yl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
3-(piperidin-4-ylmethyl)-N-[3-(pyridin-3-yloxy)propyl]benzamide
4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-2-propyl-1,3-thiazole
N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[1,2-a]pyridine-3-carboxamide
2-[4-(acetamidomethyl)piperidin-1-yl]-2-(5-fluoro-2-methoxyphenyl)acetic acid
5-cyclopropyl-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-N-[3-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
1-[(3,5-dichloro-2-methoxyphenyl)methyl]-N,N-dimethylazepan-4-amine
(1S,5R)-3-[2-(benzyloxy)ethyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-{methyl[(3-methylthiophen-2-yl)methyl]amino}pyrimidin-4-yl)piperidin-3-ol
1-methyl-6-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine-1-carbonyl)-1H-indole
(3S,4R)-1-(1-methylpiperidin-4-yl)-4-phenylpyrrolidine-3-carboxylic acid
4-benzyl-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(3-chloro-4-fluoro-1-benzothiophene-2-carbonyl)-4-(1H-imidazol-1-ylmethyl)piperidine
(1S,5R)-3-[(4-fluorophenyl)methyl]-6-(furan-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(1H-1,3-benzodiazol-1-ylmethyl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1,3-oxazole-4-carboxamide
3-(2-ethylbutyl)-8-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(azepane-1-carbonyl)-N-[2-(1H-imidazol-4-yl)ethyl]benzene-1-sulfonamide
(4aR,8aR)-2-(1-benzothiophen-2-ylmethyl)-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
3-(3-methylthiophene-2-carbonyl)-1-[(2,4,5-trimethoxyphenyl)methyl]piperidine
(2R,3R,6R)-5-[(4-ethoxyphenyl)methyl]-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-[(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)oxy]-N-(pyridin-2-ylmethyl)benzamide
8-[2-(1H-indazol-3-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
3-ethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-indole-2-carboxamide
N-ethyl-N-(1-{3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propanoyl}pyrrolidin-3-yl)acetamide
2-(1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl)pyridine
(7R,8aS)-7-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-[5-(1H-1,3-benzodiazol-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-N-cyclopentylpropanamide
1-[(3aR,6aR)-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-(4-fluorophenoxy)piperidine
2-[(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)amino]-N-ethylpyridine-4-carboxamide
8-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-cyano-N-[(3R,4S)-1-(2-methylpyridin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
propan-2-yl 4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carboxylate
4-[2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-1-(3,5-dimethylphenyl)piperazin-2-one