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1-[(2,3-difluorophenyl)methyl]-4-{1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-3-yl}piperidine
[3-(4-methylphenyl)propyl](oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
3,5-dihydroxy-N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-4-methylbenzamide
2-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1-methyl-1H-indole
(4aR,7aS)-1-methyl-4-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(4-chlorophenyl)methyl]-N-(3-ethoxy-2-hydroxypropyl)-1H-1,2,3-triazole-4-carboxamide
2-({[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}amino)pyridine-3-carbonitrile
2-{1-[(2-ethoxyphenyl)methyl]-4-[(4-ethynylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-methyl-N-{[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-1,2,3,4-tetrahydronaphthalen-1-amine
N-(morpholin-2-ylmethyl)-1-(propan-2-yl)piperidine-4-carboxamide
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-3-[(propan-2-yl)sulfamoyl]-5-[(thian-4-yl)amino]benzamide
4-chloro-1-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-pyrrole-2-carboxamide
5-{[4-(4-fluorophenyl)-1,4-diazepan-1-yl]methyl}-2,1,3-benzoxadiazole
2-[2-methoxy-6-({3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)phenoxy]propanoic acid
1-[(3-fluoro-4-methoxyphenyl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
7-(4-methylphenyl)-4-(1-propyl-1H-pyrazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}-2,3,5,6-tetramethylbenzamide
N2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-N4,N4,5-trimethylpyrimidine-2,4-diamine
2-chloro-4-({[1-(cyclohex-1-en-1-yl)ethyl]carbamoyl}amino)benzamide
[4-fluoro-3-(2,3,4-trimethoxyphenyl)phenyl]methanamine
3-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]propanamide
1-(6-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-sulfonyl}-1,2,3,4-tetrahydroquinolin-1-yl)ethan-1-one
[1-(3,3-diphenylpiperidine-1-carbonyl)cyclopropyl]methanol
2-methoxy-1-{4-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
(1S,5R)-3-benzoyl-6-(5-ethylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
N-(isoquinolin-5-ylmethyl)-N-methyl-5-propyl-1,3,4-oxadiazole-2-carboxamide
(4aS,8aS)-2-(2-amino-6-methylpyrimidin-4-yl)-decahydroisoquinolin-4a-ol
[2-(5,7-difluoro-2-methyl-1H-indol-3-yl)ethyl][1-(1H-imidazol-1-yl)propan-2-yl]amine
3-(2-hydroxyphenyl)-N-(2-methoxyethyl)-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-[1-(propan-2-yl)piperidin-4-yl]-2,9-diazaspiro[5.5]undecan-3-one
1,5-dimethyl-4-({methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
1-(1-{5H,6H-benzo[h]quinazolin-2-yl}-5-(methoxymethyl)-1H-pyrazole-4-carbonyl)-4-(2-methoxyethyl)piperazine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]propanamide
N-{2-[2-(2-methylpropyl)-6-oxo-1,6-dihydropyrimidin-4-yl]ethyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(4-fluorophenyl)-1,4-diazepane
(2S)-N-[3-(2-methoxybenzamido)phenyl]-5-oxopyrrolidine-2-carboxamide
2-(butylsulfanyl)-6-[3-(methoxymethyl)pyrrolidin-1-yl]pyrimidin-4-amine
(3aR,6aR)-2-(2-methoxyethyl)-5-(5-methyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2,3,5-trimethyl-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
3-[4-methyl-2-(oxan-2-ylmethyl)phenyl]-1,3-oxazolidin-2-one
N-{[2-(4-chlorophenyl)-5,8-dimethoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-2H-1,3-benzodioxole-5-carboxamide
1-cyclopropyl-N-(furan-2-ylmethyl)-N-[2-(morpholin-4-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(4-chloro-2-methylbenzoyl)pyrrolidin-3-yl]methanol
2-methoxy-N-[3-methyl-1-(7-{[4-(methylsulfanyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)butyl]acetamide
N-(1-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
4-(4-butoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
(4aS,8aR)-1-(3-hydroxypropyl)-6-[2-(pyridin-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-cyclopropanecarbonyl-4-{4-[4-(methoxymethyl)piperidine-1-carbonyl]phenoxy}piperidine
ethyl 2-[({3-[2-hydroxy-3-(4-methyl-1,4-diazepan-1-yl)propoxy]-4-methoxyphenyl}methyl)(methyl)amino]acetate