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N-[4-(pyridin-2-yl)butyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
2-({[2-(2-ethoxyphenoxy)ethyl](methyl)amino}methyl)-4-fluorophenol
6-{3-[3-(4-chlorobenzoyl)piperidin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
2-[(1-{[2-(dimethylamino)ethyl](methyl)amino}hex-5-en-2-yl)oxy]-N,N,5-trimethylpyrimidin-4-amine
N-methyl-N-(pyridin-3-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
1-(2-methylpropyl)-2-{[3-(pyridin-4-yl)azetidin-1-yl]methyl}-1H-1,3-benzodiazole
2-[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidine
(2S)-2-acetamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-3-(1H-imidazol-4-yl)propanamide
3-{2-[4-(3-methoxyphenyl)-2-methyl-3-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1,3-thiazole-4-carboxamide
5-methyl-3-[3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazol-5-yl]-4,5,6,7-tetrahydro-2H-indazole
(4S)-4-(propan-2-yl)-3-(quinolin-2-ylmethyl)-1,3-oxazolidin-2-one
2-(2-hydroxyphenoxy)-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-[3-(2-propoxyphenyl)propyl]oxolane-3-carboxamide
1-[4-(pyridin-4-yl)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
8-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}-1-oxa-8-azaspiro[4.5]decane
1'-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{4-[(8-fluoroquinolin-2-yl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
N-{[3-(difluoromethoxy)phenyl]methyl}-4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-(3-fluorophenyl)-N-[3-(morpholin-4-yl)propyl]-1,2,4-triazin-3-amine
1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
3-{1-[4-(morpholin-4-yl)benzoyl]piperidin-3-yl}benzoic acid
N-[1-(pyrazin-2-yl)propan-2-yl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
1-[(2-fluorophenyl)methyl]-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,4-diazepane
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-cyclopentyl-1-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(2R,3S,6R)-5-[3-(1H-imidazol-1-yl)propyl]-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(1R,3S)-1,3-dihydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(trimethyl-1H-pyrazol-1-yl)propan-1-one
(3aS,7aR)-2-[6-amino-2-(dimethylamino)pyrimidin-4-yl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-butyl-N-[(2-fluorophenyl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-(6-{4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}pyridin-3-yl)ethan-1-one
4-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1-(2-methoxyphenyl)piperazin-2-one
1-ethyl-4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
1-(5-methylthiophene-2-carbonyl)-4-(piperidine-1-sulfonyl)-1,4-diazepane
N-(1-benzylpyrrolidin-3-yl)-5-methyl-1,3,4-oxadiazol-2-amine
1'-(2H-1,3-benzodioxol-5-ylmethyl)-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4,6-dimethyl-3-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-chloro-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-5-(trifluoromethyl)benzamide
2-(dimethylamino)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]benzamide
1-(furan-2-ylmethyl)-4-[3-(propoxymethyl)pyrrolidine-1-carbonyl]piperidine
5-methyl-4-[(2-methyl-1H-imidazol-1-yl)methyl]-2-[3-(trifluoromethyl)phenyl]-1,3-oxazole
N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
7-(2-benzyl-3-oxopiperazine-1-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-3-one
(2R,3R,6R)-3-(4-fluorophenyl)-5-(4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
9-(2-hydroxyethyl)-1-methyl-4-[2-(2H-1,2,3-triazol-2-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[2-(4-fluorophenoxy)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide