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4-[6-(2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carbonyl]-2-ethyl-1-(propan-2-yl)piperazine
4-[(4-fluorophenyl)methyl]-1-[(2-phenyl-1,3-thiazol-5-yl)methyl]-1,4-diazepan-5-one
1-[9-methoxy-7-(8-methoxy-4-methylquinolin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(thiophen-3-yl)ethan-1-one
1-ethyl-8-[(3-methoxyphenyl)methyl]-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(1H-indole-6-carbonyl)-9-methoxy-N-methyl-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3S,4S)-1-[(3-hydroxyphenyl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-(propan-2-yl)-N-(pyridin-4-ylmethyl)-1,3-oxazole-4-carboxamide
1-cyclopentyl-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxamide
4-(3-methoxyphenyl)-2-(5-methyl-4-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1H-pyrazol-1-yl)pyrimidine
1-(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-4-(1H-imidazol-1-yl)butan-1-one
4-(3,4-diethoxyphenyl)-2-ethyl-1H-imidazole
N,3,6-trimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
methyl 6-({methyl[1-(thiophen-2-yl)ethyl]amino}methyl)-3-(2-phenoxyacetamido)thieno[2,3-b]pyridine-2-carboxylate
(1-{1-[1-(2-fluorophenyl)piperidin-4-yl]piperidin-3-yl}piperidin-4-yl)methanol
4-{5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
1-[2-methoxy-5-({[(5-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1-[1-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)-2-phenylethyl]-1H-1,2,3,4-tetrazole
(3-{[1-(2-phenylbenzoyl)pyrrolidin-3-yl]methyl}phenyl)methanol
benzyl 3-[2-(1H-1,2,3,4-tetrazol-5-yl)benzamido]pyrrolidine-1-carboxylate
2-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}pyrazine
7-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
N-(carbamoylmethyl)-2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-[(dimethylamino)methyl]-1-{2-methylthieno[3,2-d]pyrimidin-4-yl}azepan-4-ol
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[3-(2,5-dimethylphenoxy)propyl]-N-methylacetamide
2-methoxy-5-{[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}benzoic acid
4-[(3,4,5-trifluorophenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
5-{[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}pyrimidin-2-amine
4-{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-(piperidin-1-ylmethyl)-4-(2-propyl-1,3-thiazole-4-carbonyl)-1,4-oxazepane
2-(5-acetylthiophen-3-yl)-N-{[1-(morpholin-4-yl)cycloheptyl]methyl}acetamide
ethyl 2-(1-{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)acetate
3-[2-(morpholin-4-yl)ethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
8-cyclopentanecarbonyl-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
4-[3-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]-5,6-dimethyl-2-(trifluoromethyl)pyrimidine
4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[2-(thiophen-3-yl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-[2-(2-chloro-4-methylphenoxy)ethyl]-1,3-diazinane-2,4-dione
1-(4-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}thiophen-2-yl)ethan-1-one
1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
1-(2-aminoethyl)-N-[1-(2,4-dimethylphenyl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-cyclobutanecarbonyl-N-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]piperidine-4-carboxamide
N-(1H-imidazol-2-ylmethyl)-1-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}piperidin-4-amine
N-[3-(3-chlorophenyl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-4-carboxamide
7,8-dimethyl-3-[2-(1-methylpiperidin-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
7,8-dimethyl-2-(pyrimidin-5-yl)-4-[4-(trifluoromethyl)piperidine-1-carbonyl]quinoline
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{[7-fluoro-2-(4-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-2-(thiophen-3-yl)acetamide
(2S,4R)-1-(2,3-dihydro-1H-inden-2-yl)-4-[(4-ethylcyclohexyl)amino]-N-methylpyrrolidine-2-carboxamide
1-{2-[3-(3-chlorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-4-ethylpiperazine-2,3-dione