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3-(cyclopropylmethyl)-5-(3,5-dimethoxyphenyl)-1-methyl-1H-1,2,4-triazole
4-(4-methylpiperazin-1-yl)-6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrimidin-2-amine
2-({cyclopropyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-6-methoxyphenol
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-2,3-dimethylquinoxaline-6-carboxamide
3-(4-methyl-1H-imidazol-5-yl)-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
{[1-(2-methoxyethyl)piperidin-4-yl]methyl}(methyl)(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)amine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[2-(2,3-dimethylphenoxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(cyclopropylmethyl)-5-[4-methyl-2-(propan-2-yl)pyrimidine-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methylbenzamide
2-(3-phenylpiperidin-1-yl)-N-(thiophen-2-ylmethyl)acetamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}thiophene-2-carboxamide
1-{5-[3-(2-phenylethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-4-ol
N-[(1S,2S)-2-[(4-fluorophenyl)methyl]cyclopentyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
2-(phenylamino)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}pyrimidine-5-carboxamide
N-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-5-(5-methylfuran-2-yl)-1,2,4-triazin-3-amine
N-[2-(2,5-dimethylphenoxy)ethyl]-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}-N-methylacetamide
5-{[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
2-[2-methyl-3-({[(3-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1H-indol-1-yl]acetamide
N-[2-(4-methoxyphenyl)ethyl]-N-[(1-methylpiperidin-4-yl)methyl]-6-oxo-1,6-dihydropyrimidine-5-carboxamide
5-cyclopropyl-1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-N-(1-methoxybutan-2-yl)-1H-pyrazole-4-carboxamide
methyl({2-[2-(prop-2-en-1-yl)phenoxy]ethyl})(pyridin-4-ylmethyl)amine
2-[4-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-1-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
1-[3-(2,2-dimethylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-[(5-methyl-1H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
1-methanesulfonyl-4-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1,4-diazepane
1-ethyl-1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3-(1,2,3-thiadiazol-5-yl)urea
2-methyl-4-phenyl-5-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]pyrimidine
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-3-methylpiperidine
N4-(furan-2-ylmethyl)-N1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)piperidine-1,4-dicarboxamide
3-(1H-imidazol-2-yl)-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
2-[4-(4-cyclohexylpiperazine-1-carbonyl)-5-cyclopropyl-1H-pyrazol-1-yl]-4-(2-fluorophenyl)pyrimidine
4-{[1,2,4]triazolo[4,3-a]pyrazin-3-yl}quinoline
7-(2,2-dimethylpropyl)-2-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
5-{5-[2-(1-methylpiperidin-3-yl)ethyl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
7-[(2,3-difluorophenyl)methyl]-2-(3-methylbut-2-en-1-yl)-2,7-diazaspiro[4.5]decane
2-(adamantan-1-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide
2-[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]-N-(5-fluoro-2-methylphenyl)acetamide
6-(propan-2-yl)-3-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
4-methyl-2-oxo-5-[3-(piperidin-1-ylmethyl)piperidine-1-carbonyl]-1,2-dihydropyridine-3-carbonitrile
[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-4-yl](thiophen-2-yl)methanol
1-(4-fluorophenyl)-5-{[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-1H-1,2,4-triazole
4,6-dimethyl-1-{2-[4-(oxolan-3-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
3-methyl-N-{2-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]ethyl}thiophene-2-carboxamide
N-(furan-2-ylmethyl)-N-(thiophen-2-ylmethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
(1R,5R)-N,N-dimethyl-6-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl]ethane-1-sulfonamide
ethyl 2-{methyl[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]amino}-1,3-oxazole-4-carboxylate
2-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
N,N-diethyl-1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxamide
4-[5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carbonyl]-2-(trifluoromethyl)morpholine