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N-cyclohexyl-N-methyl-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
2-(5-acetylthiophen-3-yl)-1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
methyl(2-phenylethyl){[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}amine
N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-[(4-phenoxyphenyl)methyl]acetamide
[4-(3,4-dichlorophenyl)pyridin-2-yl]methanol
2-[5-(2-cyclopropyl-4-methylpyrimidin-5-yl)-1-(2,3-dimethylphenyl)-1H-1,2,4-triazol-3-yl]acetamide
(4aS,8aR)-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
4-(3-hydroxy-3-methylbutyl)-N-methyl-N-(oxan-2-ylmethyl)benzamide
2-(2,4-dichlorophenoxy)-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}acetamide
2-(4-methoxy-3-methylphenyl)-4-(3-methyl-1,2,4-oxadiazol-5-yl)pyridine
3-{3-[({2-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}amino)methyl]-1H-indol-1-yl}propanamide
4-{[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]methyl}-N-methylbenzene-1-sulfonamide
1-(2-hydroxy-3-{4-[(4-hydroxypiperidin-1-yl)methyl]-2-methoxyphenoxy}propyl)piperidin-4-ol
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-ethyl-1H-1,2,4-triazole
N-[(2-chlorophenyl)methyl]-3-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]propanamide
(4aS,8aR)-6-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
(3S,4R)-1-(2-fluorobenzoyl)-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
N-[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4,4,4-trifluorobutanamide
4-{2-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamido]ethyl}benzoic acid
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]pyridazine-4-carboxamide
6-methyl-2-{1-[(4-methyl-1H-imidazol-5-yl)methyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}-5,5-diphenylpiperidin-2-one
4-{1-[1-(1,2-oxazole-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
ethyl 5-[(4-methoxyphenyl)methyl]-1-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-(2-hydroxyethyl)-9-(2-methoxy-4-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
6-(2-methoxyphenyl)-N-methyl-N-(pyrimidin-4-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2,7-diazaspiro[4.5]decane
2-(cyclopentylmethyl)-N-(2-hydroxy-2-phenylethyl)-N,6-dimethyl-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(thiophen-2-ylmethyl)amino]methyl}piperidin-2-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-5-methoxyfuran-2-carboxamide
5-[1,3-dimethyl-5-(morpholin-4-yl)-1H-pyrazol-4-yl]-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-2-methyl-1H-1,3-benzodiazole-5-carboxamide
[3-(cyclopropylmethyl)-1-(furan-3-ylmethyl)piperidin-3-yl]methanol
7-(4-fluorobenzoyl)-N-(1-methoxypropan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-ethyl-4-[5-(2-methylphenyl)-4-phenyl-1H-imidazol-1-yl]piperidine-1-carboxamide
1-ethyl-4-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl}ethan-1-ol
1-(dimethyl-1,2-oxazole-4-carbonyl)-3-(3-methylphenoxymethyl)piperidine
4-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-7-chloro-4-methylquinolin-2-amine
1-[3-(1H-pyrazol-1-yl)benzoyl]-4-(pyridin-2-ylmethyl)-1,4-diazepane
{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(methyl)[1-(pyridin-2-yl)propan-2-yl]amine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-6-azaspiro[2.5]octane-1-carboxamide
2-({[(3R,4R)-1-(3-chloro-2-methylbenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
9-(8-hydroxy-5,7-dimethylquinoline-2-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-({1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}amino)-4,6-dimethylpyridine-3-carbonitrile