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N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
3-({2-[3-(1H-indol-3-yl)-1-methyl-1H-1,2,4-triazol-5-yl]ethyl}(methyl)amino)-1λ6-thiolane-1,1-dione
N-(4-phenyl-1,2,3-thiadiazol-5-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide
5-[3-(piperidine-1-carbonyl)pyridin-2-yl]quinoline
(2S)-2-{[5-(4-cyclohexylphenyl)-1,2,4-triazin-3-yl]amino}-4-(methylsulfanyl)butan-1-ol
1-ethyl-5-oxo-N-[6-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]pyrrolidine-3-carboxamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-pyrrole-2-carboxamide
1-{4-[(furan-2-ylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
3-[benzyl({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amino]propanamide
5-ethyl-2-(1-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1H-imidazol-2-yl)pyridine
7-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N-(2-phenylphenyl)-4-[2-(pyrrolidin-1-yl)ethyl]piperazine-1-carboxamide
2-(1H-indazol-1-yl)-1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
9-(5-methyl-1H-indazole-3-carbonyl)-1,4,9-triazaspiro[5.5]undecan-5-one
N-(3,5-dimethoxyphenyl)-2-{[(1R)-2-hydroxy-1-phenylethyl]amino}acetamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
2-benzyl-4-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]morpholine
N-(furan-2-ylmethyl)-1-[(4-methylphenyl)methyl]-5-oxo-N-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
4-(2-{3-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}ethyl)morpholine
4-fluoro-3-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}benzene-1-sulfonamide
4-(2-fluoro-5-methylphenoxy)-1-(pyridine-4-carbonyl)piperidine-4-carboxylic acid
3-hydroxy-1-(2-methoxyethyl)-3-{[4-(pyrazin-2-yl)piperazin-1-yl]methyl}piperidin-2-one
N-{2-[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}acetamide
methyl({[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl})(thiophen-3-ylmethyl)amine
4-[7-(3-methylfuran-2-carbonyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrrolidine-1-carboxamide
(1R,5S,8R)-8-(dimethylamino)-N-{4-[(2-methylprop-2-en-1-yl)oxy]phenyl}-3-azabicyclo[3.2.1]octane-3-carboxamide
1-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
6-phenyl-3-{1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-1,2-dihydropyridin-2-one
[(4S)-4-amino-5-[4-(2-chlorophenoxy)piperidin-1-yl]-5-oxopentyl]urea
3-{4-[4-phenyl-1-(pyridin-2-ylmethyl)-1H-imidazol-5-yl]phenyl}prop-2-yn-1-ol
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]acetamide
2-methyl-6-{1-oxa-8-azaspiro[4.6]undecane-8-carbonyl}-2,3-dihydropyridazin-3-one
2-oxo-N-propyl-N-(pyridin-3-ylmethyl)-2H-chromene-3-carboxamide
2-(pyridin-3-yl)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
7-methyl-3-{[methyl(pyrazin-2-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
1-({4-methyl-5-[1-(1-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)azepane
(3aS,6aR)-5-(6-methoxypyrimidin-4-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-[4-(4-methanesulfonylphenyl)phenyl]-2-(morpholin-4-yl)ethan-1-ol
methyl 2-{[5-(cyclooctylcarbamoyl)-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridin-3-yl]formamido}acetate
5-{2-methylimidazo[1,2-a]pyridin-6-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-(2,3-dihydro-1H-inden-2-yl)-N-propyloxane-4-carboxamide
1-[(3-fluorophenyl)methyl]-4-(6-methylquinolin-4-yl)piperazin-2-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-{spiro[indene-1,4'-piperidine]-1'-yl}ethan-1-one
{2-[2-(1-{imidazo[1,2-a]pyridine-3-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
7-(3-chlorophenyl)-4-(5-methoxyfuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(3-hydroxyphenyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]propanamide
1-(2,6-difluoro-3-methylbenzoyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol